13/308,658
`
`drug potency
`drug selectivity
`drug synthesis
`ITLOUSS
`
`*non insulin dependent diabetes mellitus
`nonhuman
`
`CT
`
`*structure activity relation
`Drug Descriptors:
`a og'
`iptin: AN, drug ana;ysis
`a'og'ipti n: P
`D, pharmaco;ogy
`*azo;opyrimidine: AN, drug ana;ysis
`*azo;opyrimidine:
`PD, pharmaco;ogy
`*dipeptidy;
`peptidase IV inhibitor: AN, drug ana;ysis
`*dipeptidy; P
`eptidase IV inhibitor:
`PD, pharmaco;ogy
`inag'
`iptin.
`AN, drug ana;ysis
`'inag'
`iptin:
`PD, pharmaco;ogy
`saxag;iptin:
`AN, drug ana;ysis
`saxag;iptin:
`PD, pharmaco;ogy
`sitag;iptin:
`AN, drug ana;ysis
`sitag;iptin:
`PD, pharmaco;ogy
`unc;assified drug
`'iptin: AN, drug ana;ysis
`'iptin:
`PD, pharmaco;ogy
`DPP4; GLP-1; SAR
`Azo;opyrimidines;
`Iogliptin) 850649-61-5;
`(1inag;iptin)
`Q\: _.\ .\-
`,\
`Nfiffifim
`I
`babuus
`as1£sg~0§~8
`“~i;
`(sitag;iptin)
`) 27490l—l6—5
`
`668270—12—0;
`486460-32-6,
`
`(vi;dag1iptin
`
`(saxagliptin)
`65467l—78—0;
`
`=> fi
`1e s
`:nguide
`FI.?
`«N T«%«D AT 09:19:55 ON 01
`'STNGUID* .'
`_AY 2012
`-1
`.«M
`TO
`Tin TnRMS Ob YOUR CUSTO
`USE I
`S SU?J?CT
`«R AGR
`
`CO
`?YRIGHT
`_A ERICAN CHTMICAL SOCITTY
`2012
`(C)
`CHARG
`33 TO COST=TC1600
`
`(ACS)
`
`fiNT
`
`FI.?
`LAST
`
`CONTAINS CURRENT INFORMATION.
`
`RnLOAD«D: Apr 27, 2012 (20120427/UP).
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:25)(cid:20)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-IPRZO16-01104- Ex. 1006. Part 2, p. 161 of 373
`
`291
`
`0420
`0420
`
`

`
`13/308,658
`
`=> d his ful
`
`CHARG
`
`(t1..
`ED TO
`
`«NT«
`'HOM«'
`COST=TC160
`
`«D AT 08:07:49 ON 01 MAY 2012)
`
`«R
`
`«NT
`'ZCAP.JS'
`COST=TC16OO
`E US2001-788173/APPS
`
`«D AT 08:08:08 ON 01 MAY 2012
`
`FITF‘.
`CHARG
`ED TO
`
`FILE
`CHARG
`ED TO
`L1
`
`«R
`
`«NT
`'HCAPLJS'
`COST=TC16OO
`1 S«A S?
`D SCAN
`3EL L1 1-
`
`«D AT 08:08:26 ON 01 MAY 2012
`
`«=ON A33=ON
`
`PLU=ON US2001-788173/APPS
`
`RN
`
`«D AT 08:08:42 ON 01 MAY 2012
`
`OOOOOO/U/U/U/U/U/U/U
`
`1
`
`1 1
`
`«NT «R
`t1L«
`'R«G1ST3Y'
`CHARG
`ED TO COST=TC16OO
`PLU=ON
`L2
`242 S«A S?«=ON A33=ON
`31 OR 102502-64-7/31
`(1000689-56-4/
`OR 102507-13-1/31
`OR 104757-47-3/31 OR 1
`05-53-3/31 OR 1068-90-2
`31 OR
`/31 OR 108-94-1/3
`1 OR 1098535-00-2/
`31 OR 1098535-01-3/
`OR
`OR
`1098535-02-4/31
`1098535-03-5/31
`1098535-04-6/31
`OR
`OR
`1098535-05-7/31
`1098535-06-8/31
`1098535-07-9/31
`OR
`OR
`1098535-08-0/31
`1098535-09-1/31
`1098535-10-4/31
`OR
`OR
`1098535-11-5/31
`1098535-12-6/31
`1098535-13-7/31
`OR
`OR
`1098535-14-8/31
`1098535-15-9/31
`1098535-16-0/31
`OR
`OR
`1098535-17-1/31
`1098535-18-2/31
`1098535-19-3/31
`OR
`OR
`1098535-20-6/31 O
`1098535-21-7/31
`1098535-22-8/31
`31 O
`1098535-23-9/31 OR
`1098535-24-0/31 OR 11
`91-95-31
`R 120-92-3/
`31 OR 13031-04-4/3
`OR 13139-16-7/
`31 OR 13433-00-6/31 OR
`13837-45-1/31 OR
`14328-51-9/
`31 OR 143979-40-2/31 OR 144643-84-5
`31 OR 144978-12-1/31 OR 15023-45-7/
`31 OR 1576-87-0/31 OR
`31 OR 1781
`31 OR 179015-57
`73724-30-6/31 OR
`173724—34-0/
`72-26-41
`-7/31 OR 179
`015-58-8/
`31 OR 18928—91—11
`31 OR 1903-22-6/31 OR
`31 OR 200424-69-
`191655-45-5/31 OR
`19550-72-2/
`31 OR l97l42—36—2/
`7/31 OR 20859-02-3
`
`'/31
`OR 2094-74-8/
`31 OR 2130-96-3/31 OR
`31 OR 2141
`31 OR 21573-69-
`214193-10-9/31 OR 211
`193-11-01
`93-13-2/
`31
`3/31 OR 2356-16-3/
`OR 2534-90-9/31 O
`R 3005-66-1/31 OR
`4
`31 OR 3614
`31 OR 361440-62-
`35264-06-3/31 OR 36111
`0-58-61
`0-61—1/
`31 OR
`31 OR 361
`2/31 OR 361440-63-3/31 OR 361440-64-4/
`140-65-51
`31 OR 361440-70
`361440-66-6/31 OR 3611
`40-67-71
`31 OR 361440-69-9/
`31 OR
`31 OR 361
`-2/31 OR 361440-71-3/31 OR 361
`440-73-51
`440-77-91
`31 OR 3614
`31 OR 361440-91
`361440-78-0/31 OR 3611
`40-79-11
`40-88-21
`31 OR
`31 OR 361
`-7/31 OR 361440-95-1/31 OR 361
`440-97-31
`440-99-51
`31 OR 3614
`31 OR 361441-05
`361441-01-2/31 OR 3611
`41-03-41
`41-04-51
`31 OR
`31 OR 361
`-6/31 OR 361441-06-7/31 OR 361
`441-07-81
`441-08-91
`41-10-3131 OR 3614
`31 OR 361441-12
`361441-09-0/31 OR 3611
`41-11-41
`31
`31 OR 361
`-5/31 OR 361441-13-6/31 OR 361441-14-7/
`441-15-81
`I)
`_ _4U=ON
`150 S «A SP«=ON A33=ON
`'
`L2 AND C3-NC4/ES
`
`L3
`
`t1L«
`'LR«G1STRY'
`CHARG
`ED TO COST=TC16OO
`L4
`STR
`
`«NT«R
`
`«D AT 08:10:11 ON 01 MAY 2012
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:25)(cid:21)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-|PR2016-01104- Ex. 1006. Part 2, p. 162 of 373
`
`292
`
`0421
`0421
`
`

`
`13/308,658
`
`nNTnRnD AT 08:15:03 ON 01 MAY 2012
`tILn 'RnGIST3Y'
`CHARGED TO COST=TC1600
`L5
`50 SEA SSS SA
`
`L4
`
`tILn 'LRnGISTRY'
`CHARGED TO COST=TC1600
`L6
`STR L4
`
`nNTn3nD AT 08:15:38 ON 01 MAY 2012
`
`nNTnRnD AT 08:16:15 ON 01 MAY 2012
`tILm 'RnGIST3Y'
`CHARGED TO COST=TC1600
`L7
`50 SEA SSS SA
`
`L6
`
`nVTn3nD AT 08:16:57 ON 01 MAY 2012
`FI.E 'STVGUIDn'
`CHARGED TO COST=TC1600
`
`tI.n 'LRnGIST3Y'
`CHARGED TO COST=TC1600
`L8
`STR L6
`
`nNTn3nD AT 08:17:39 ON 01 MAY 2012
`
`nNTnRnD AT 08:17:51 ON 01 MAY 2012
`tILn 'RnGIST3Y'
`CHARGED TO COST=TC1600
`L9
`50 SEA SSS SA
`
`L8
`
`"121 |—|
`nWTn3nD AT 08:18:53 ON 01
`'STNGUIDn'
`"E
`CHARGED TO COST=TC1600
`
`.AY 2012
`
`nVTn3nD AT 08:19:58 ON 01
`tlun 'RnGIST3Y'
`CHARGED TO COST=TC1600
`
`.AY 2012
`
`tI.n 'L3nGISTRY'
`CHARGED TO COST=TC1600
`L10
`STR L8
`
`nNTn3nD AT 08:20:31 ON 01 MAY 2012
`
`nNTnRnD AT 08:21:03 ON 01 MAY 2012
`tILn 'RnGIST3Y'
`CHARGED TO COST=TC1600
`L11
`50 SEA SSS SA
`
`L10
`
`nNTnRnD AT 08:21:56 ON 01 MAY 2012
`FILE 'STNGUIDn'
`CHARGED TO COST=TC1600
`D QUE S TAT
`
`tILn 'LRnGISTRY'
`CHARGED TO COST=TC1600
`L12
`STR L10
`
`nNTnRnD AT 08:28:12 ON 01 MAY 2012
`
`nNTnRnD AT 08:29:43 ON 01 MAY 2012
`tILn 'RnGIST3Y'
`CHARGED TO COST=TC1600
`L13
`50 SEA SSS SA
`
`L12
`
`nNTnRnD AT 08:30:11 ON 01 MAY 2012
`FILE 'STNGUIDn'
`CHARGED TO COST=TC1600
`D QUE S TAT
`
`tILn 'RnGISTRY'
`
`nNTnRnD AT 08:32:40 ON 01 MAY 2012
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:25)(cid:22)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-IPR2016-01104- Ex. 1006. Part 2, p. 163 of 373
`
`293
`
`0422
`0422
`
`

`
`13/308,658
`
`CHARGED TO COST=TC1600
`E14
`8057 SEA SSS FJE L12
`SAVE TEMP
`.14 ?OL658PSET1/A
`15 SEA S?t=ON A33=ON PLJ=ON
`D SCAN
`
`E15
`
`L3
`
`L14
`
`«NT.%nD AT 08:33:40 ON
`FI.E 'STNGUIDn'
`CHARGED TO COST=TC1600
`
`01
`
`_AY
`
`2012
`
`nNT.%nD AT 08:35:08 ON
`tlun 'RnGIST%Y'
`CHARGED TO COST=TC1600
`L16
`135 SEA S?t=ON A33=ON PLU=ON
`
`01
`
`_AY
`
`2012
`
`L2
`
`AND
`
`L14
`
`
`.
`FI.?
`.«NT .%ED AT 08:35:23 ON
`'STWGUID*'
`CHARGED TO COST=TC1600
`
`01
`
`MAY
`
`2012
`
`11.E 'LREGISTRY'
`CHARGED To CoST=TC1600
`L17
`STR
`
`ENTERED AT 08:38:02 ON 01 MAY 2012
`
`ED AT 08:41:44 ON 01 MAY 2012
`
`TILE 'REGIST%Y' ENTER
`CHARGED To CoST=TC1600
`E18
`0 SEA SJS=.14 SSS SAM E17
`D QJE STAT
`4 SEA SJ3=.14 SSS FUL E17
`SAVE TEM? L19 RoL658NSET1/A
`D SCAN
`
`E19
`
`TILE 'LREGISTRY' ENTERED AT 08:44:15 ON 01 MAY 2012
`CHARGED To CoST=TC1600
`L20
`STR L12
`
`«D AT 08:46:21 ON 01 MAY 2012
`
`L22 NOT L19
`
`TILE 'REGIST%Y' ENTER
`CHARGED To CoST=TC1600
`E21
`50 SEA SJS=.14 SSS SAM E20
`D QJE STAT
`8057 SEA S 3=.14 SSS FUL E20
`SAVE TEM?
`.22 ?O.658%SET1/A
`8053 SEA S?E=oN A33=oN
`?LJ=ON
`SAVE TEM?
`.23 ?o.658CRoSS/A
`D SC N L19
`
`E22
`
`E23
`
`FILE 'STNGUIDE' ENTER
`CHARGED To COST=TCl6OO
`D SAVED
`
`ED AT 08:48:55 ON 01 MAY 2012
`
`FILE 'ZCAPLUS' ENTERED AT 08:49:36 ON
`CHARGED To COST=TCl6OO
`E24
`QUE S?E=oN AES=oN PEU=oN
`E25
`QUE S?E=oN A33=oN PEU=oN
`E26
`QUE S?E=oN A33=oN PEU=oN
`E27
`QUE S?E=oN AES=oN PEU=oN
`E28
`QUE S?E=oN A33=oN PEU=oN
`E29
`QUE S?E=oN A33=oN PEU=oN
`
`01
`
`_AY 2012
`
`ROE
`I,
`J?/AU,AUTH,IN
`SUE
`SKY,
`‘H,IN
`R?/AU,AUt
`SUE
`SKY,
`‘H,IN
`D?/AU,AUt
`AUG
`ER1,
`‘H,IN
`D?/AU,AUt
`MAG
`NIN,
`‘H,IN
`D?/AU,AUt
`HAMANN, L?/AU,AUt
`‘H,IN
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:25)(cid:23)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-IPRZO16-01104- Ex. 1006. Part 2, p. 164 of 373
`
`294
`
`0423
`0423
`
`

`
`13/308,658
`
`L30
`
`QUE SPE=ON ARR=ON
`
`PLU=ON
`
`RETERENNER, D?/AU,AUTH,IN
`
`FILE 'HCAPLUS' ENTERED AT 08:50:44 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`PLU=ON
`L31
`1 SEA SPE=ON ARR=ON
`OR L28 OR L29 OR L30)
`D RI?
`
`L1 AND (L24 OR L25 OR L26 OR L27
`
`FILE 'ZCAPLUS' ENTERED AT 08:51:00 O\ 01 MAY 2012
`CHARGED TO COST=TC1600
`
`L32
`
`QUE S?E=ON ARR=ON
`MY<2001 OR REVIEW/DT
`
`PLU=O\ AY<2001 OR PY<2001 OR PRY<2001 OR
`
`FILE 'HCAPLUS' ENTERED AT 08:51:58 O\ 01 MAY 2012
`CHARGED TO COST=TC1600
`PEU=O\
`E33
`725 SEA S?E=ON ARR=ON
`PEU=O\
`E34
`26 SEA S?E=ON ARR=ON
`OR L28 OR L29 OR L30)
`0 SEA S?E=ON ARR=ON
`PEU=O\
`26 SEA S?E=ON ARR=ON
`PEU=O\
`699 SEA S?E=ON ARR=ON
`PEU=O\
`142 SEA S?E=ON ARR=ON
`PEU=O\
`
`E35
`E36
`E37
`E38
`
`E23
`E33 AND (L24 OR L25 OR L26 OR L27
`
`E1 NOT L34
`(L34 OR E35)
`E33 NOT E36
`E37 AND E32
`
`FI.E 'STNGUIDE' ENTERED AT 08:53:26 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`
`tI.E 'LREGISTRY' ENTERED AT 08:55:08 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`L39
`STR L12
`
`EILE 'REGISTRY' ENTERED AT 08:55:41 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`L40
`50 SEA SJR=.14 SSS SAM L39
`
`FILE 'STNGUIDE' ENTERED AT 08:56:21 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`D QUE S ‘TAT
`
`tILE 'REGISTRY' ENTERED AT 08:59:05 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`E41
`6632 SEA SJR=.14 SSS FUL L39
`SAVE TEM?
`.41 ?Ou658NSET2/A
`1421 SEA S?*=ON ARR=ON
`PLJ=ON L23 NOT L41
`SAVE T*M3
`.42 ?Ou658CROSS2/A
`
`E42
`
`FILE 'STNGUIDE' ENTERED AT 09:00:19 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`D SAVED
`
`FI.E 'HCAPLUS' ENTERED AT 09:00:54 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`
`tI.E 'REGISTRY' ENTERED AT 09:01:03 ON 01 MAY 2012
`CHARGED TO COST=TC1600
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:25)(cid:24)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-IPRZO16-01104- Ex. 1006. Part 2, p. 165 of 373
`
`295
`
`0424
`0424
`
`

`
`13/308,658
`
`27 SEA S?E=ON ARR=ON
`
`PLU=ON
`
`L16 NOT L42
`
`FILE 'HcARLUS' ENTERED AT 09:02:03 ON 01 MAY 2012
`ARG
`ED TO cOST=Tc1600
`427 SEA S?E=ON ARR=ON
`
`PLU=ON
`
`L42
`
`
`
`LLLLLLOv\v\v\v\l\l\"|"
`
`U‘InJ>
`
`Q)(X)\10‘\
`
`RLU=ON
`15 SEA S?E=ON ARR=ON
`OR L28 OR L29 OR L30)
`0 SEA S?E=ON ARR=ON
`RLU=ON
`15 SEA S?E=ON ARR=ON
`RLU=ON
`412 SEA S?E=ON ARR=ON
`RLU=ON
`87 SEA S?E=ON ARR=ON
`RLU=ON
`
`L44 AND (L24 OR L25 OR L26 OR L27
`
`L1 NOT L45
`(L45 OR L46)
`L44 NOT L47
`L48 AND L32
`
`II.E 'REGISTRY' ENTERED AT 09:03:44 ON 01 MAY 2012
`CPARG
`ED TO cOST=Tc1600
`
`FI.E 'HcARLUS' ENTERED AT 09:03:55 ON 01 MAY 2012
`CPARG
`ED TO cOST=Tc160
`L50
`TRA ?LJ=ON L49 1- RN HIT
`
`74 TERMS
`
`CHARG
`_J5].
`_J52
`
`L53
`
`IILE 'REGISTRY' ENTERED AT 09:04:00 ON 01 MAY 2012
`ED TO cOST=Tc1600
`74 SEA S?E=ON ARR=ON
`74 SEA S?E=ON ARR=ON
`E SAXAGLI?TIN/CN
`1 SEA S?E=ON ARR=ON
`3 SCAN
`
`RLU=ON
`RLU=ON
`
`L50
`L51 NOT L2
`
`RLU=ON
`
`SAXAGLIRTIN/CN
`
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`icicicicicicicicicicicicicicic
`
`J:IT.E 'HOME'
`
`EN
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`TERED AT 15:43:05 ON 30 APR 2012
`
`=> fil reg
`
`J:I .E
`.N~n
`'REGISTRY
`TO Ti
`USE IS S
`JRJECT
`PLEASE S
`EE "HEPP USAGE
`
`RED AT 15:43:22 ON 30 APR 2012
`4
`TERMS Ob YOUR STN
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`I"! 4IRMS I!
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`v
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`CO?YRIG{T (C) 2012 American Chemical
`
`Society
`
`(ACS)
`
`Property values tagged with IC are
`provided by InfoChem.
`3.
`1
`E J:IT..
`UPDAT
`AS
`RY FI
`E UPDATE
`
`from
`
`the ZIC/VINITI data file
`
`HIGH
`HIGH
`
`L‘J U)
`L‘J U)
`
`‘I
`F RN 1371145-50-4
`‘I
`F RN 1371145-50-4
`
`STRUCTUR
`DICTIONA
`
`:
`S:
`
`29 APR 2012
`29 APR 2012
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:26)(cid:22)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-|PR2016-01104- Ex. 1006. Part 2, p. 173 of 373
`
`303
`
`0432
`0432
`
`

`
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`TSCA INFORMATION NOW CURRENT THROUGH DECEMEER 23, 2011
`
`Please note that search—term pricing does apply when
`conducting SmartSELECT searches.
`
`REGISTRY includes nimerica"y searchable data for experimental and
`predicted properties as we" as tags indicating availability of
`experimental proper:y data in the original document.
`For information
`on property searching in REGISTRY, refer to:
`
`
`
`*** YOU HAVE NEW MAI. ***
`
`=> s saxagliptin/cn
`L1
`1 SAXAGEIPTIN/CN
`
`=> d 11
`
`El
`RN
`ED
`
`ANSWER 1 Oh
`361442-O4-8
`Entered STN:
`
`I
`
`REGISTRY COPYRIGHT 2012 ACS on STN
`REGISTRY
`11 Oct 2001
`
`CN
`
`2—Azabicyclo[3.1.0]heXane—3—carbonitrile,
`2—[(28)—2—amino—2—(3—hydroxytricyclo[3.3.1.13,7]dec—1—yl)acetyl]—,
`(lS,3S,5S)-
`(CA INDEX NAME)
`OTHER CA INDEX NAMES:
`
`CN
`
`(1S,3S,5S)-
`
`2—Azabicyclo[3.1.0]heXane—3—carbonitrile,
`2—[(28)—amino(3—hydroxytricyclo[3.3.1.13,7]dec—1—yl)acetyl]-,
`(9CI)
`OTHER NAMES:
`CN
`3M8 477118
`CN
`3M8 477118-11
`CN
`CN
`FS
`DR
`MF
`CI
`SR
`
`
`
`.
`_.
`1339955—48—4
`C18 {25 N3 O2
`CO
`CA
`
`LC
`
`CENR, CHEMCATS,
`ADISINSIGHT, AVABSTR, CA, CAPLUS, CASREACT
`STV Files:
`IPA, MRCK*,
`CHEMLIST, DDFU, DRUGU, EMEASE,
`IMSPATENTS,
`IMSRESEARCH,
`?ATDPASPC, PS, RTECS*, TOXCEVTER, USAW, USPAT2, USPATFULE
`(*File contains numerically searchable proper:y data)
`
`I
`
`Absolute stereochemistry.
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:26)(cid:23)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-IPR2016-01104- Ex. 1006. Part 2, p. 174 of 373
`
`304
`
`0433
`0433
`
`

`
`HO
`
`CN
`
`S
`
`N
`
`S
`
`**PROR
`
`ERTY DATA AVAI.A%LE IN THE '?RO?' FORMAT**
`
`-—..
`4)
`IVES
`
`1 1
`
`313 RntnRnNCfiS IN tI.n CA (1907 TO DAC
`IN tILL; CA
`4 RntnRnNCnS TO NON—SPLCIfIC DERIVAC
`330 RntnRnNCfiS IN tI.n CAPLUS
`(1907 TO DATE)
`
`=> s saxagliptin
`L2
`5 SAXAGLIPTIN
`
`=> d l2 1-
`
`YOU HAVn %nQUnSTnD DATA FROM 5 ANSWERS - CONTINUE? Y/(N):y
`
`E2
`RN
`
`ANSWER 1 Or
`945667-22-1
`
`5
`
`REGISTRY COPYRIGHT 2012 ACS on STN
`REGISTRY
`
`«D
`CN
`
`28 Aug 2007
`«ntered STN:
`2—Azabicyc;o[3.l.0]heXane—3—carbonitrile,
`2—[(28)—2—amino—2—(3—hydroxytricyclo[3.3.l.l3,7]dec—l—yl)acetyl]—, hydrate
`(1:1),
`(1S,3S,5S)-
`(CA INDnX NAMn)
`OTHnR NAMnS'
`
`CN
`FS
`MF
`SR
`
`LC
`
`CRN
`
`
`Saxa» gtin hy§1.ta
`ST*.R*.OS*.ARCH
`H2 O
`C18 {25 N3 O2
`CAS Client Services
`
`nMEASfi,
`ADISIWSIGHT, CA, CAPLUS, CASREACT, CHEMCATS,
`STN Files:
`IMSRnSnARCH,
`IPA, MRCK*, TOXCnNTnR,
`JSAN, US?AT2, USPATFULL
`IMSPATENTS,
`(*File contains numerically searchable Orooerty data)
`(36l442—04—8)
`
`Absolute stereochemistry.
`
`s
`
`s
`
`o
`
`C>H2o
`
`**PROPERTY DATA AVAILA EH
`
`-11
`
`-144
`
`IN TH
`
`‘PROP’ FORMAT**
`
`(cid:54)(cid:88)(cid:81)(cid:16)(cid:36)(cid:80)(cid:81)(cid:72)(cid:68)(cid:79)(cid:16)(cid:44)(cid:51)(cid:53)(cid:21)(cid:19)(cid:20)(cid:25)(cid:16)(cid:19)(cid:20)(cid:20)(cid:19)(cid:23)(cid:16)(cid:3)(cid:40)(cid:91)(cid:17)(cid:3)(cid:20)(cid:19)(cid:19)(cid:25)(cid:17)(cid:3)(cid:51)(cid:68)(cid:85)(cid:87)(cid:3)(cid:21)(cid:15)(cid:3)(cid:83)(cid:17)(cid:3)(cid:20)(cid:26)(cid:24)(cid:3)(cid:82)(cid:73)(cid:3)(cid:22)(cid:26)(cid:22)
`Sun-Amneal-|PR2016-01104- Ex. 1006. Part 2, p. 175 of 373
`
`305
`
`0434
`0434
`
`

`
`ntnR nNC ES IN tI m
`3 R
`3 R ntnR nNC ES IN tI a
`
`CA
`(1907 TO DATE
`)
`CAPLUS
`(1907 TO DAT
`
`E2
`RN
`«D
`
`ANSWER 2 Or
`841302-24-7
`«ntered STN:
`
`5
`
`REGISTRY COPYRIGHT 2012 ACS on STN
`REGISTRY
`03 Mar 2005
`
`CN
`
`2—Azabicyc1o[3.1.0]heXane—3—carbonitri;e,
`_o[3.3.1.13,7]dec—1—y1)acety1]—,
`2
`[(28)
`2 amino 2
`(3,5 dihydroxytricyci
`(1S,3S,5S)-
`(CA INDnX NAMn)
`OTHER CA INDnX NAMnS:
`
`2—Azabicyc1o[3.1.0]heXane—3—ca