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`EXAMINER IN CHIEF
`
`U.S. PATENT AND TRADEMARK OFFICE
`RETURN TO
`Interference Service Branch
`This case is involved in an
`Interference Proceeding.
`
`PTO»1058
`
`INTERFERENCE
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`Sawai Ex 1005
`Page 1 of 4322
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`

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`Sawai Ex 1005
`Page 2 of 4322
`
`

`
`hiJ of
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`FORM PT0-650
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`M." HK OFFICE .
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`! i d i rrRJjCbb
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`INTERFERENCE—INITIAL MEMORANDUM
`EXAMINERS INSTRUCTIONS-^—This ,form need not be typewritten. Complete the items below and forward to the Group Clerk with all
`files deluding those benefit of which has been accorded. The parties need nortiepis^^in
`specific
`order. Use a separate form for each count.
`•
`
`(See MPEP 2309.02)
`
`BOARD OF PATENT APPEALS AND INTERFERENCES: An Interference is found to exist between the following cases:
`
`\ This is count
`
`of
`
`count{s).
`
`AME
`
`SERIAL NO.
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`FILING DATE
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`The claims of this party which correspond to this count are;
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`PATENT NO., IF ANY _
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`The claims of this party which correspond to this count are:
`The claims of this party which do not correspond to this cpunt
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`DATE
`PRIMARY EXAMINER
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`Clerk's instructions:
`1. Obtain a title report for all cases and include a copy.
`2. Forward all files including those benefit of which is being accorded.
`
`/"$
`
`0
`
`Sawai Ex 1005
`Page 3 of 4322
`
`

`
`BOARD SMSSr0""*-"1
`INTERFERENCE—INITIAL MEMORANDUM,PPEALS &
`
`TRADEMARK OFFICE
`
`mhm)
`
`>OflM PTO-850
`(REV 3-86)
`
`ip Clerk with all
`EXAMINERS INSTRUCTIONS—This .form need not be typewritten. Complete the items below aifd
`isted in any specific
`rded. The parti^pe^i not be^li
`files including those benefit of which has been acco
`order. Use a separate form for each count.
`
`(See MPEP 2309.02)
`
`IARD OF PATENT APPEALS AND INTERFERENCES: An Interference Is found to exist between the following cases:
`
`This is count
`
`of
`
`count(s)
`
`SERIAL NO.
`
`FILING DATE
`
`PATENT NO., IF ANY
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`1. HIKME
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`he claims of this party which correspond to this count ar&
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`
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`SERIAL NO.
`
`FILING DATE
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`PATENT NO.. IF ANY
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`^ I The claims of this party which do not correspond to "fnis count
`are:
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`7//33.57 6
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`\ SERIAL NO.
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`The claims of this party which correspond to this couni are^
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`The ctaims of this pariy which do not correspond to fhrp'Sjsunr
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`The claims of this party which correspond to this count are:
`
`FILING DATE
`
`3 - >3-90
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`The claims of this party which do not correspond to this count
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`If a claim of any party is exactly the same as this count, it should be circled above. If not. type the count in this space ijattacirot^fit^l .
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`DATE
`PRIMARY EXAMINER
`fca-o-qi
`
`'
`Clerk's instructions:
`1. Obtain a title report for all ceses and include a copy.
`2. Forward all files including those benefit of which is being accorded.
`
`GROUP DIRECTOR SIGNATURE.(if required)
`
`La
`
`be listed.
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`
`Sawai Ex 1005
`Page 4 of 4322
`
`

`
`' ••ffW.IO'.'^'IF" J 1 r*—
`
`in"!
`
`*
`
`FORM PT0-850
`{R£V. 3-86)
`
`INTERFERENCE—INITIAL MEMORANDUM
`
`u's. DEPARTMENT OF COMMERCt
`PATENT AND TRADEMARK OFFICE
`
`m
`
`EXAMINERS INSTRUCTIONS—This form need not be typewritten. Complete the items below and forward to the Group Clerk with all
`files including those benefit of which has been accorded. The parties need not be listed in any specific
`.
`order. Use a separate form for each count.
`'
`'•
`
`(See MPEP 2309.02)
`
`OARD OF PATENT APPEALS AND INTERFERENCES: An Interference is found to exist between the following cases:
`of
`
`X
`
`count(s).
`
`X
`
`This is count
`\ I SERIAL NO,
`FILING DATE
`NAME
`t oJ' \
`12.-7-^7
`1^,516
`P l f A R N p
`The claims of this party which do not correspond to-'this-jptfjfit
`The claims of this party which correspond to this>count 3i\
`15
`© y 2 . - ^CoSoMtd)
`are:
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`ii
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`PATENT NO., IF ANY
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`COUNTRY
`
`SERIAL NO.
`
`FILING DATE
`
`2X
`
`NAME
`
`i -
`
`IAJ A I r AM A S) Mi
`The claims of this party which correspond to this count are:
`1 (W 10
`
`t)
`
`FILING DATE
`
`l-ai-qo
`
`PATENT NO., IF ANY
`
`The claims of this pany which do not correspond to this count.
`are:
`
`• Accorded benefit of:
`COUNTRY
`'
`
`its.
`
`SERIAL NO.
`Q7/ 3 I ^ 7 7 ^
`
`FILING DATE
`
`3-7'^
`
`PATENT NO., IF ANY
`
`3. .NAME
`
`SERiALNO.
`
`FILING DATE
`
`PATENT NO., IF ANY
`
`The claims of this party which correspond to this count are:
`
`The claims of this party which do not correspond to this count
`are:
`
`* Accorded benefit of:
`COUNTRY
`
`SERIALNO.
`
`FILING DATE
`
`PATENT NO., IF ANY
`
`If a claim of any party is exactly the same as this count, it should be circled above. If not; type the count in this space (attach additional
`sheet if necessary}:
`"
`
`vft
`
`'
`
`•
`
`' The serial number and filing date of each application the benefit of which is intended to be accorded must be listed. It is not sufficient to
`merely list the earliest application if there are intervening applications necessary for continuity.
`DATE
`
`PRIMARY EXAMINER
`
`i - a j - q i
`
`JrthMOiO
`
`'
`Clerk's instructions:
`1. Obtain a title report for all cases and include a copy.
`2. Forward all files including those benefit of which is being accorded.
`
`TELEPHONE NO/
`
`wr-^s-jz-
`
`ART UNIT
`
`I 2 D I
`
`GROUP DIRECTOR SIGNATURE (if required)
`
`Sawai Ex 1005
`Page 5 of 4322
`
`

`
`FORM PTO-850
`IR6V. 3-86)
`
`(See MPEP 2309.02)
`
`INTERFERENCE—INITIAL MEMORANDUM
`EXAMINERS INSTRUCTIONS—This jorm need not be typewritten. Complete the items below and forward to the Group Clerk with all
`files fpcluding those benefit of which has been accorded. The parties need not be listed in any specific
`.order. Use a separate form for each count.
`•
`
`U.S. DEPARTMENT OF COMMERCE
`PATENT AND TRADEMARK OFFICE
`
`BOARD OF PATENT APPEALS AND INTERFERENCES: An Interference is found to exist between the following eases:
`
`This is count ^ of ^ count(s).
`A
`\
`'
`XNAME
`SERIAL NO.
`-filrod ^
`^
`The claims of this party which correspond to this count ar^S^
`(S) ((zMa^zJ)
`
`) - / 4
`
`FILING DATE
`
`The claims of this party which do not correspond to this count
`are:
`
`7
`
`PATENT NO., IF ANY
`
`v.na mi
`
`* Accorded benefit of:
`COUNTRY
`
`SERIAL NO.
`
`FILING DATE
`
`PATENT NO.. IF ANY
`
`/
`
`^S^NAME
`
`\Nf\- M
`
`S'/N
`
`The claims of this party which correspond to this count are:
`
`SERIAL NO.
`
`TlimOl
`
`FILING DATE
`
`1-23-10
`
`/ CD
`•
`PATENT NC£5F AN§
`:-o^ o
`' ^ £ 2
`tortji^<^t
`
`"o" SjC/JjS
`m Fffl
`^ Q ^ -HI
`to 2:
`PATENT NO.. IF ANM
`
`The claims of this party which do not corresp
`are:
`
`(.rzHouJClMc)
`^ ^
`* Accorded benefit of:
`COUNTRY
`V
`SERIAL NO.
`u-s-
`
`"4-
`
`1-7,1 0
`i-s-ry
`
`FILING DATE
`
`3. NAME
`
`SERIAL NO,
`
`FILING DATE
`
`PATENT NO.. IF ANY
`
`The claims of this party which correspond to this count are:
`
`The claims of this party which do not correspond to this count
`are:
`
`' Accorded benefit of:
`COUNTRY
`
`«
`
`SERIAL NO.
`
`FILING DATE
`
`PATENT NO.. IF ANY
`
`(f a claim of any party is exactly the same' as this count, it should be circled above. If not. type the count in this space (attach additional
`sheet if necessary):
`
`yft
`
`* The serial number and filing date of each application the benefit of which is intended to be accorded must be listed. It is not sufficient to
`merely list the earliest application if there are intervening applications necessary lor continuity.
`DATE
`PRIMARY EXAMINER
`
`00/^/0 focbfreH
`
`TELEPHONE NO:
`
`Z 0 8-liS'3:L
`
`ART UNIT
`
`no I
`
`Clerk's instructions:
`T. Obtain a title report for all cases end include a copy.
`2. Forward ail files including those benefit of which is being accorded.
`
`GROUP DIRECTOR SIGNATURE (if required)
`
`Sawai Ex 1005
`Page 6 of 4322
`
`

`
`Interference No. 102,648
`
`-1-
`
`The cases involved in this interference are:
`Junior Party
`Applicant: Sompong Wattanasin
`Address: 11 Divito Trail Hopatcong, New Jersey 07843
`07/498,301 filed 03/23/90
`Serial No.:
`For: Quinoline Analogs Of Mevalonolactone And Derivatives Thereof
`Assignees: None
`Attorneys of Record:
`
`Gerald D. Sharkin, Robert S. Honor,
`Richard E. Villa, Walter F. Jewell, Thomas
`0. McGovern, Thomas c. Doyle, Melvyn M.
`Kassenoff, Joseph J. Borovian, Joanne M.
`Giesser and Diane E. Furman
`Associate Attorney: None
`Accorded Benefit of: U.S. Serial No. 07/318,773 filed 03/03/89
`Gerald D. Sharkin
`Address:
`Sandoz Corp.
`59 Route 10
`E. Hanover, NJ 07936
`Junior Party
`Patentees: Joseph A. Piqard, Bruce D. Roth and Drago R.
`Sliskovic \
`/
`Addresses: 3545 GreenbrierVpt. 65C, Ann Arbor, Michigan 48105
`1440 King GeorgeNjlW., Ann Arbor, Michigan 48104
`4860 Cole Blvd., Y^silanti, Michigan 48197
`Serial No.: 07/129,516 filed 12/1X7/81, Patent No. 4,761,419
`issued 08/02/88
`j \
`For: 6-(((Substituted)Quinolinyl)Ethyl)-And Ethenyl)Tetrahydeo-
`4-Hydroxypyran-2-One Inhibitors>of Cholesterol Biosynthesis
`Assignees: Warner-Lambert Company, A Corp. of DE
`Attorneys of Record: Elizabeth M. Anderson^ Ronald A. Daignault,
`Charles Gaglia, Jerry IT. Janssen., Henry
`Jeanocte, Anne M. KellyV Gary M. Nath,
`Howard Olevsky, Stephen Raines, Daniel A.
`Scola and Joan Thiersteiri\
`
`r
`
`Sawai Ex 1005
`Page 7 of 4322
`
`

`
`Interference No. 102,648
`
`It
`
`Associate Attorney: None
`Accorded Benefit of: None
`Address: Jerry. F. Janssen
`WarnervrLambert Co.
`2800 pii
`iouth Road
`Ann Arb<
`, MI 48105
`Senior Party
`Applicants: Yoshihiro Fujikawa, Mikio Suzuki, Hiroshi Iwasaki,
`Mitsuaki Sakashita and Masaki Kitahara
`•
`Addresses: Nissan Chemical Industries, Ltd, Chuo Kenkyusho,
`722-1, Tsuboi-cho, Funabashi-shi, chiba-ken, Japan
`Serial No.: 07/233,752 filed 08/19/88
`.
`For: Quinoline Type Mevalonolactones
`Assignees: Nissan Chemical Industries Ltd., Tokyo, Japan
`Attorneys of Record: Norman F. Obion, Stanley P. Fisher, Marvin
`J. Spivak, C. Irvin McClelland, Gregory J.
`Maier, Arthur I. Neustadt, Robert C.
`Miller, Richard D. Kelly, James D.
`Hamilton, Eckhard H. Kuesters, Robert T.
`Pous, Charles L. Gholz, Vincent J.
`Sunderdick, William E. Beaumont and Steven
`B. Kelber
`Associate Attorney: None
`Accorded Benefit of: Japan Serial Nos. 207224 filed 08/20/87 and
`15585 filed 01/26/88
`OVa/l
`Address: Obion, Fisher, Spivak,
`McClelland & Maier
`1755 S. Jeff. Davis Hwy.
`Crystal Square 5, Ste. 400
`Arlington, VA 22202
`
`s?
`
`Sawai Ex 1005
`Page 8 of 4322
`
`

`
`Interference No. 102,648
`
`Count 1
`
`A compound of structural Formula I
`
`-3-
`
`R4.
`
`Rj
`
`RJ
`
`•.Ri
`
`N
`
`X—A
`
`R2
`
`R6
`
`wherein A is
`
`HO H
`/
`
`i ml
`
`H
`
`o ^ o
`
`*
`
`>
`
`X is —CH2CH2— or —CK=CH—;
`Rj and R2 are independently
`hydrogen;
`alkyl of from one to six carbons;
`trifluoromethyl;
`.
`cycloprdpyl;:
`.*
`cyclohexyl;
`cyclohexylmethyl;
`^
`phenyl;
`phenyl substituted with
`fluorine,
`chlorine,
`bromine,
`hydroxy,
`trifluoromethyl,
`alkyl of from one to four carbon atoms, or
`alkoxy of from one to four carbon atoms;
`phenylmethyl;
`phenylmethyl substituted with
`fluorine,
`chlorine,
`bromine,
`hydroxy,
`. trifluoromethyl,
`alkyl of from one to four carbon atoms, or
`alkoxy of from one to four carbon atoms;
`2-, 3-, or 4-pyridinyl; or
`2-, 4-, or 5-pyrimidinyl;
`
`'
`
`Sawai Ex 1005
`Page 9 of 4322
`
`

`
`Interference No. 102,648
`
`™ 4 w
`
`.
`
`Rj, R* Rj, R<s are independentiy selected from
`hydrogen;
`alky] of from one to six carbon atoms;
`trifluoromethyl;
`cyclopropyl;
`fluorine;
`chlorine;
`bromine;
`hydroxy;
`alkoxy of from one to four carbon atoms;
`cyano;
`nitro;
`amino;
`acetylamino;
`aminomethyl;
`phenyl;
`phenyl substituted with
`fluorine,
`chlorine,
`bromine,
`hydroxy,
`trifluoromethyl,
`aJkyl of from one to four carbon atoms, or
`alkoxy of from one to four carbon atoms;
`phenylmethyl; or
`phenylmethyi substituted with
`fluorine,
`chlorine,
`bromine,
`-
`hydroxy,
`.
`trifluoromethyl, or
`alkyl of from one to four carbon atoms;
`provided that when X is in the 2-position, RJ is hydro*
`gen and is attached in the 4-position;
`or a corresponding 3,5-dihydroxyacid of Formula II
`
`.
`
`Sawai Ex 1005
`Page 10 of 4322
`
`

`
`Interference No. 102,648
`
`-5-
`
`*3
`
`.*i
`
`II
`
`HO
`H 0
`^ /% / i
`X—C CHj—C—CHjCOH
`
`Rj
`
`N
`
`R:
`
`wherein A, X, Rj, Rj, R], R4, and Rj are as defined
`above, or a pharmacruticaUy acceptable salt
`thereof!
`
`The claims of the parties which correspond to Count 1
`
`are:
`Wattanasin
`Picard et al.
`Fujikawa et al.
`
`Claims 1-7 and 10
`Claims 1-14
`Claims 1-9, 11-34, 36, 39 and 40
`
`Count 2
`
`A method of inhibiting cholesterol biosynthesis in a
`patient in need of said treatment comprising administering a
`cholesterol synthesis inhibiting amount of a compound as def ined
`by count 1 in combination with pharmaceutically acceptable
`carrier.
`
`The claims of the parties which correspond to Count 2
`
`Claims 8 and 9
`Claim 15
`Claims 35, 37 and 38
`
`Michael Sbfbfclgous
`Examiner-in-Chief
`(703) 557-4066
`
`are:
`Wattanasin
`Picard et al.
`Fujikawa et al.
`
`X
`
`-
`
`Sawai Ex 1005
`Page 11 of 4322
`
`

`
`Alt coMMimMfiau raptctiag this
`am tkomid Utrntify it by numbtr
`tnd Mfliftfj qfparties.
`
`Paper No. 2
`'• V
`
`% #
`
`o*
`
`U.S. DEPARTMENT OF COMMERCE
`Parant: and Trademark Office
`
`Address: BOX INTERFERENCE
`Commissioner of Patents end Trademarks
`Washington. D.C. 20231
`(703)557-4007
`Telephone:
`(703)557-8642
`Facsimile:
`
`#
`
`MAILED
`M4R 1 1 1992
`
`Interference No. 102,648
`Wattanasin
`V.
`Picard et al.
`V.
`Fujikawa et al.
`
`This interference has been assigned to the undersigned in
`accordance with 37 CFR 1.610. All future papers filed in this
`interference should be captioned to include this information.
`Any questions regarding procedure in this interference
`should be directed to the undersigned. However, any such contact
`must include the participation of both parties, e.g., via a
`conference call.
`Each party is required to file a paper in accordance with 37
`CFR 1.613 identifying its lead attorney or agent (see 37 CFR
`1.601(3c)) by no later than 2 ji MAR 1992 . Future changes in the
`lead attorney or agent must likewise be called to the attention
`of this board as soon as reasonably possible. No contact should
`be made with the undersigned by anyone other than the lead
`attorneys or agents.
`The time for filing and serving notice of filing (but not
`serving) preliminary statements (37 CFR 1.621 - 1.628) and for
`filing preliminary motions (37 CFR 1.633, et. seq.. note in
`particular.
`1.637) is set to expire 11 .nm m?
`The parties are strongly encouraged to make contact with
`each other at the time that its lead attorney or agent are
`identified in an attempt to settle this interference. The
`examiner-in-chief can be expected to cooperate in allowing
`reasonable time for a bona fide attempt at settlement
`negotiations, which will obviate the necessity for filing
`preliminary motions and will result in the filing of an
`appropriate termination paper under 37 CFR 1.662.
`
`• •
`
`Sawai Ex 1005
`Page 12 of 4322
`
`

`
`Interference No. 102,648
`
`-2-
`
`There has been confusion regarding the use of the "BOX
`INTERFERENCE" requirement of 37 CFR 1.1(e) in the filing of
`papers. Unless the paper itself is hand carried to the Service
`Branch of the Board of Patent Appeals and Interferences, located
`in Room 10C01 of Crystal Gateway 2 (1225 Jefferson Davis Highway,
`Arlington, VA), the designation "BOX INTERFERENCE" must be on the
`outside of the envelope containing the paper as well as on the
`paper itself. Merely hand carrying a paper to the PTO Mail Room
`does not suffice.
`
`Summary of Times Running
`1. Statements and Motions due
`Identity of lead attorney or agent due
`2.
`
`1 1 JUN 199? •
`2 5 MAR 1992
`-
`
`gjh
`
`/j
`
`Michael Sofbcjfeous
`Examiner-in-Chief
`(703) 557-4066
`
`Sawai Ex 1005
`Page 13 of 4322
`
`

`
`IN THE UNITED STATES PATENT AND TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCES
`
`BOARD OF PATENT
`APPEALS *
`WTERFtf®GES
`m\i ^
`
`WATTANASIN
`V.
`PICARD ET AI*
`V.
`FUJIKAWA ET AL
`
`: INTERFERENCE 102,648
`:
`EXAMINER-IN-CHIEF :
`MICHAEL SOFOCLEOUS
`I
`:
`
`•
`
`PESIGNATTnw nv r.g&n rnnwfiEL, 37 CFR Sl,601(k)
`
`HONORABLE COMMISSIONER OF PATENTS AND TRADEMARKS
`WASHINGTON, DC 20231
`BOX INTERFERENCE
`
`SIR:
`Pursuant to 37 CFR §l,601(k), the Senior Party Fujikawa et al
`hereby designates as lead attorney Steven B., Kelber, Reg. No.
`30,0731.
`
`Respectfully submitted,
`QBLON, SPIVAK, McCLELLAND,
`MAIER & NEUSTADT, P.C..
`
`\
`Steven B. Kelber
`Registration No•:
`Attorney of Record 30,073
`Fourth Floor
`1755 South Jefferson Davis Highway
`Arlington, Virginia 22202
`703-521-5940
`
`Sawai Ex 1005
`Page 14 of 4322
`
`

`
`CERTIFICATE OP SERVICE
`
`I hereby certify that true copies of:
`
`DESIGNATION OF LEAD COUNSEL, 37 CFR §1.601(k)
`
`were served upon Counsel for the Wattanasin and Picard et al as
`follows:
`
`and
`
`Gerald D. Sharkin, Esq.
`Sandoz Corp.
`59 Route 10
`E. Hanover/ NJ 07936
`
`Jerry F. Janssen, Esq.
`Warner-Lambert Co.
`2800 Plymouth Road
`Ann Arbor, MI 48105
`
`via first-class mail, postage prepaid, this 17th day of March,
`1992.
`
`STEVEN B. KELBER
`
`Sawai Ex 1005
`Page 15 of 4322
`
`

`
`IN THE UNITED STATES PATENT AND TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCES
`
`WATTANA5IN
`V,
`PICARD ET AL
`V.
`FUJIKAWA ET AL
`
`INTERFERENCE 102,648
`EXAMINER-IN-CHIEF :
`MICHAEL SOFOCLEOUS
`
`-r -
`
`O
`OS
`
`2:
`
`^rn0
`-n
`-o
`
`CO 3:
`
`00
`
`?s
`
`POWER TO INSPECT AMD MAKE COPIES
`
`BOX INTERFERENCE
`HONORABLE COMMISSIONER OF PATENTS AND TRADEMARKS
`WASHINGTON, DC 20231
`SIR:
`The undersigned, being an Attorney of Record for the above-
`identified Interference, hereby grants to MURALIDHAR PAI/SAM BROWN,
`the power to inspect and make copies of the above-identified
`Interference files.
`
`Respectfully submitted,
`OBLON, SPIVAK, KcCLELLAND,
`MAIE;
`NEUST.
`P.C.
`A
`Steven B. Kelber
`Registration No.:
`Attorney of Record 30,073
`
`' 'V
`
`Sawai Ex 1005
`Page 16 of 4322
`
`

`
`BOARD OF PATENT
`APPEALS &
`WTERFERENCES
`IN THE UNITED STATES PATENT AND TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCES
`26 1992
`
`WATTANASIN
`V*
`PICARD ET AL
`V.
`FUJIKAWA ET AL
`
`INTERFERENCE 102,648
`EXAMINER-IN-CHIEF :
`MICHAEL SOFOCLEOUS
`
`SUPPLEMENTAL
`DESIGNATTnw OF T.igiir> COUNSEL. 37 CFR Sl.601fkl
`
`HONORABLE COMMISSIONER OF PATENTS AND TRADEMARKS
`WASHINGTON, DC 20231
`BOX INTERFERENCE
`
`SIR:
`Superseding Senior Party Fujikawa's earlier filed Designation
`of Lead Counsel, 37 CFR §1.601(k) is a Supplemental Designation of
`Lead Counsel, 37 CFR §1.60l(k) correctly identifying Lead Counsel's
`Registration Number as 30,073. The Senior Party Fujikawa regrets
`this inadvertent error and any inconvenience it may have caused.
`Respectfully submitted,
`OBLON, SPIVAK, McCLELLAND,
`MAIER & NEUSTADT, P.C.
`
`Steven B. Kelber
`Registration No.:
`Attorney of Record
`Fourth Floor
`1755 South Jefferson Davis Highway
`Arlington, Virginia 22202
`703-521-5940
`
`30,073
`
`Sawai Ex 1005
`Page 17 of 4322
`
`

`
`BOARD OF PATENT
`APPEALS &
`INTERFERENCES
`IN THE UNITED STATES PATENT AND TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCE 26 1992
`
`WAXTANASIN
`V.
`PICARD ET AL
`V.
`FUJIKAWA ET AL
`
`INTERFERENCE 102,648
`EXAMINER- IN-CHIEF :
`MICHAEL SOFOCLEOUS
`
`SUPPLEMENTAL
`PESIGNATT<""J OP T.BAP COUNSEL, 37 CFR Sl.SOlfkl
`
`HONORABLE COMMISSIONER OF PATENTS AND TRADEMARKS
`WASHINGTON, DC 20231
`BOX INTERFERENCE
`
`SIR:
`Pursuant to 37 CFR Sl.SOlfk)/ the Senior Party Fujikawa et al
`hereby designates as lead attorney Steven B. Kelber, Reg. No.
`30,073.
`
`Respectfully submitted,
`.OBLON, SPIVAK, McCLELLAND,
`MAIER & NEUSTADT, P.C.
`
`Fourth Floor
`1755 South Jefferson Davis Highway
`Arlington, Virginia 22202
`703-521-5940
`
`Steven B. Kelber
`Registration No.:
`Attorney of Record 30,073
`
`• '»
`
`Sawai Ex 1005
`Page 18 of 4322
`
`

`
`CERTIFICATE OF SERVICE
`
`I hereby certify that true copies of:
`
`SUPPLEMENTAL DESIGNATION OF LEAD COUNSEL, 37 CFR §1.601(k)
`
`were served upon Counsel for the Wattanasin and Picard et al as
`follows;
`
`and
`
`Gerald D. Sharkin, Esq.
`Sandoz Corp.
`59 Route 10
`E. Hanover, NJ 07936
`
`Jerry F. Janssen, Esq.
`Warner-Lambert Co.
`2800 Plymouth Road
`Ann Arbor, MI 48105
`
`via first-class mail, postage prepaid, this 26th day of March,
`1992.
`
`S1
`
`:N B. KELBER
`
`Sawai Ex 1005
`Page 19 of 4322
`
`

`
`Case No. 600-7101/CONT
`Patent
`MAR 25 1992
`IN THE UNITED STATES PATENT AND TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AMD INTERFERENCES SOX l«TfRFffi£|VC£
`
`RECEH'ED IN
`
`•„ FYf
`
`WATTANASIN
`v.
`PICARD et al.
`v.
`FUJIKAWA et al.
`
`Interference No. 102,648
`Examiner-in-Chief:
`M. Sofocleous
`
`Honorable Commissioner of Patents and Trademarks
`Washington, D.C.
`20231
`BOX INTERFERENCE
`37 CFR 1.602 NOTIFICATION OF INTEREST
`FOR THE PARTY WATTANASIN
`
`In accordance with 37 CFR 1.602, the Board of Patent
`Appeals and Interferences is hereby advised that the involved
`application of the party Wattanasin is assigned to, and the
`real party in interest is, Sandoz Pharmaceuticals Corpora­
`tion, a corporation of Delaware, having its principal place
`of business at 59 Route 10, East Hanover, New Jersey 07936.
`
`Respectfully submitted.
`
`Jfant
`Shljll-
`Diane E. Furman
`Attorney for the Party Wattanasin
`Registration No. 31,104
`201-503-7332 (phone)
`201-503T8807 (facsimile)
`
`I hereby otrtify that 1MB eerrMpondane* it being
`deporttad with tht Unittd Stttat Poatal Service w
`first dew meM In •* envelope eddressed to: Ctommte-
`•toner cf RNMi MtWMMmton. OC.
`20231,
`JU
`e E. Fnrman _
`.
`m
`ML
`
`SANDOZ CORP.
`59 Route 10
`E. Hanover, NJ 07936
`RMF:def
`March 24, 1992
`
`Sawai Ex 1005
`Page 20 of 4322
`
`

`
`CERTIFICATE OF SERVICE
`
`It is hereby certified that true copies of the paper
`entitied:
`
`37 CFR 1.602 NOTIFICATION OF INTEREST
`FOR THE PARTY WATTANASIN
`
`were served on counsel for the parties Fujikawa et al. and
`Picard et al., this 24th day of March, 1992, by postage pre­
`paid first-class mail addressed to the following:
`
`Warner-Lambert Co.
`Patent Department
`Attn: Jerry F. Janssen, Esq.
`2800 Plymouth Road
`Ann Arbor, MI 48105
`for the party Picard et al.
`
`Obion, Spivak, McClelland, Maier & Neustadt, P.C.
`Attn: Steven B. Kelber, Esq.
`1755 South Jefferson Davis Highway
`Crystal Square 5, Ste. 400
`Arlington, VA 22202
`for the party Fujikawa et al.
`
`MM*
`Diane E. Furman
`
`2
`
`Sawai Ex 1005
`Page 21 of 4322
`
`

`
`\
`ANV
`
`S' «c 'iA
`
`Case No. 600-7101/CONT
`Patent
`Uu THE UNITED STATES PATENT AMD TRADEMARK OFFICE
`
`EilfrORB THE BOARD OF PATENT APPEALS AND INTERFERENCES ^7
`
`WATTANASIN
`v.
`PICARD et al.
`v.
`FUJIKAWA et al.
`
`Interference No. 102,648
`Examiner-in-Chief:
`M. Sofocleous
`
`=3
`
`M-,.
`> ^3 i-J ft"
`O ^ rn rr;
`CO
`
`Honorable Commissioner of Patents and Trademarks
`20231
`Washington, D.C.
`BOX INTERFERENCE
`
`37 CFR 1.613 DESIGNATION OF LEAD ATTORNEY
`FOR THE PARTY WATTANASIN
`
`In accordance with 37 CFR 1.613, the undersigned, =Diane
`'•v
`E. Furman, is hereby designated as the lead attorney for the
`party Wattanasin in the above-identified interference.
`Melvyn M. Kassenoff, Registration No. 26,389, attorney
`of record at phone no. (201) 503-8477, is hereby designated
`deputy lead attorney with full power and authority to act in
`the absence, for any reason, of the lead attorney.
`As per the power of record, the address for both of the
`foregoing
`is: Patent and Trademark Department, Sandoz
`Corporation, 59 Route 10, East Hanover, New Jersey 07936.
`
`I hereby certify that this correspondence is being
`deposited with the United States Postal Servicers
`first class mail in an envelope addressed to: Commis­
`sioner of Patents and Tredemarka, Washington, D.C.
`a*231-" Marfih 33, 199?,,
`Diane i!^¥u¥n§n
`pfajDsScanT
`or
`Ive
`1ML
`MarBff83, 1992
`Date of SIg nature
`SANDOZ CORP.
`59 Route 10
`E. Hanover, NJ 07936
`RMFsdef
`March 23, 1992
`
`Respectfully submitted,
`
`'fkunA/x^
`
`Diane E. Furman
`Attorney for the Party Wattanasin
`Registration No. 31,104
`201-503-7332 (phone)
`201-503-8807 (facsimile)
`
`Sawai Ex 1005
`Page 22 of 4322
`
`

`
`4/
`
`^ MAR 24
`39
`
`tt*
`
`CERTIFICATE OF SERVICE
`
`V-f,*
`
`It is hereby certified that true copies of the paper
`entitled:
`
`37 CFR 1.613 DESIGNATION OF LEAD ATTORNEY
`FOR THE PARTY WATTANASIN
`
`were served on counsel for the parties Fujikawa et al. and
`Picard et al., this 23rd day of March, 1992, by postage pre­
`paid first-class mail addressed to the following:
`
`Warner-Lambert Co.
`Patent Department
`Attn: Jerry F. Janssen, Esq.
`2800 Plymouth Road
`Ann Arbor, MI 48105
`for the party Picard et al.
`
`Obion, Spivak, McClelland, Maier & Neustadt, P.C.
`Attn: Steven B. Kelber, Esq.
`1755 South Jefferson Davis Highway
`Crystal Square 5, Ste. 400
`Arlington, VA 22202
`for the party Fujikawa et al.
`
`3 fft—
`/jfiUtb
`Diane E. Furman
`
`- 2
`
`Sawai Ex 1005
`Page 23 of 4322
`
`

`
`CD
`S O
`' =5 m > S
`zo Ig o
`• "nmQ
`rr\
`CN -y j>
`-T\
`rn i o
`^3 ^ co >
`--o ho m m
`O J?o I
`oo .
`
`PATENT
`CASE NO. 600-7101/CONT.
`
`IN THE UNITED STATES PATENT AMD TRADEMARK OFFICE
`
`In ReJ SOMPONG WATTANASIN
`Serial No.: 07/498,301
`Filed: March 23, 1990
`For:
`QUINOLINE ANALOGS OF MEVALONOLACTONE AND DERIVATIVES
`THEREOF
`
`POWER TO INSPECT AND MAKE COPIES
`
`Honorable Cominissioner of
`Patents and Trademarks
`Washington, D.C. 20231
`
`. Dear Sir:
`
`Kindly permit Marian Schwartz, Ann Rutledge, Rosalie
`Jared, Somchay Chinyavong, Judy Valusek, James Jackson, Bobbie
`Judy, or Nancy Perry of Specialized Patent Services to inspect and
`make copies in the above noted matter, including recently declared
`Interference No. 102,648 in which said patent is involved.
`
`SANDOZ CORP.
`59 Route 10
`E. Hanover, N.J. 07936
`
`DEFJIcr
`
`April 1,.1992
`
`End.: postcard
`
`Respectfully submitted.
`
`Y&ftg
`By.
`(AVMCun-
`Diane E. Furman
`Registration No. 31,104
`(201) 503-7332
`
`"I/I /?£.
`
`Sawai Ex 1005
`Page 24 of 4322
`
`

`
`IN THE UNITED STATES PATENT & TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCES
`
`Wattanasin
`v.
`Picard, et al.
`v.
`Fujikawa, et al.
`
`+
`
`Interference No. 102,648
`Examiner-In-Chief:
`Michael Sofocleous
`
`FYI
`
`+
`
`^ 1992
`RECEIVED IN
`DOX INTERFERENCE
`DESIGNATION OF LEAD ATTORNEY
`FOR THE PARTY PICARD, ET AL.
`
`BOX INTERFERENCE
`Hon. Commissioner of Patents and Trademarks
`Washington, D.C. 20231
`Sir:
`The party Picard, et al. hereby designates RONALD A.
`DAIGNAULT, Registration Number 25,968, as lead attorney for the
`above-identified interference,
`The lead attorney's address and
`direct dial telephone are:
`
`WARNER-LAMBERT COMPANY
`2800 Plymouth Road
`Ann Arbor, MI 48105
`(313) 996-7530
`
`Dated:
`
`/ffZ-
`/
`
`Respectfully submitted.
`
`Ronald
`. Daignault
`Registration No. 25,968
`Attorney for the party
`Picard, et al.
`
`RAD:cm/184/3
`
`Sawai Ex 1005
`Page 25 of 4322
`
`

`
`PROOF OF SERVICE UNDER 37 C.g.R. §1.646 AND
`CERTIFICATE OF MAILING UNDER 37 C.F.R. Sl»8(a)
`
`I hereby state that true and complete copies of the
`DESIGNATION OF LEAD ATTORNEY FOR THE PARTY PICABD, ET AL. was
`served upon the parties Wattanasin and Fujikawa, et al. this 6th
`day of April, 1992, by mailing same with sufficient first class
`postage affixed and prepaid as follows:
`
`For the Party Wattanasin
`Diane E. Furman, Esq.
`SANDOZ CORP.
`59 Route 10
`East Hanover, NJ 07936
`
`and
`
`For the Party Fujikawa, et al.
`Steven B. Kelber, Esq.
`OBLON, SPIVAK, McCLELLAND,
`MAIER & NEUSTADT, P.C.
`Fourth Floor
`1755 S. Jefferson Davis Hwy.
`Arlington, VA 22202
`
`Furthermore, I hereby certify that this correspondence is
`being deposited today with the United States Postal Service with
`sufficient postage as first class mail in an envelope addressed
`to:
`Commissioner of Patents and Trademarks, BOX INTERFERENCE,
`Washington, D.C. 20231.
`
`Dated th
`
`C , r f f i r -
`f
`
`Ronald A. 'Dai&nault
`(Reg. No. 25,968)
`
`1
`
`Sawai Ex 1005
`Page 26 of 4322
`
`

`
`IN THE UNITED STATES PATENT & TRADEMARK OFFICE
`BEFORE THE BOARD OF PATENT APPEALS AND INTERFERENCES
`#10
`Interference No. 102,648
`Examiner-In-Chief:
`Michael Sofocleous
`FYI
`
`+
`
`Wattanasin
`V.
`Picard, et al.
`v.
`Fujikawa, et al.
`
`+
`
`1992
`RECEIVED IN
`BOX INTERFERENCE
`
`REQUEST BY THE PARTY PICARD, ET AL.
`UNDER 37 CFR 1.662(a) FOR
`ENTRY OF ADVERSE JUDGMENT AS TO
`COUNTS 1 AND 2 OF THE INTERFERENCE
`
`BOX INTERFERENCE
`Hon. Commissioner of Patents and Trademarks
`Washington, D.C. 20231
`Sir:
`The party Picard, et al. hereby requests entry of Adverse
`Judgment as to the subject matter of Counts 1 and 2 of the
`Interference which corresponds to Picard, et al.'s Claims 1 and
`•
`2-14.
`
`Respectfully submitted.
`
`£,
`Dated:
`Warner-Lambert Company
`2800 Plymouth Road
`Ann Arbor, MI 48105
`
`t
`
`Ronald A. Daign;
`It
`Registration No. 25,968
`Attorney for the party
`Picard, et al.
`
`RAD:cm/183/3
`
`Sawai Ex 1005
`Page 27 of 4322
`
`

`
`PROOF OF SERVICE UNDER 37 C.F.R. §1.646 AND
`CERTIFICATE OF MAILING UNDER 37 C.F.R. S1.8£a)
`
`I hereby state that true and complete copies of the
`REQUEST BY THE PARTY PICARD, ET AL. UNDER 37 CF