`First Disintegrant
`Water Soluble Excipient
`Water Soluble Polymer Binder
`Granule
`
`5-40 mg; select 10 mg
`5-300%
`250-2000%
`6-80%
`
`Second disintegrant
`Total mass
`
`20-1200% of granule
`
`WITHOUT % lurasidone
`LUBRICANT % first disintegrant
`% water soluble excipient
`% water soluble polymer binder
`% second disintegrant
`
`Optional lubricant
`Total mass with lubricant
`
`0.3 to 3% of total tablet
`
`% lurasidone
`WITH
`LUBRICANT % first disintegrant
`% water soluble excipient
`% water soluble polymer binder
`% second disintegrant
`% lubricant
`
`API
`
`max
`
`min
`
`10
`0.5
`25
`0.6
`36.1
`
`10
`30
`200
`8
`248
`
`7.22
`43.32
`
`2976
`3224
`
`23.08%
`
`0.31%
`
`0.13
`43.45
`
`96.72
`3320.72
`
`23.01%
`
`0.30%
`
`First Disintegrant
`max
`min
`
`10
`30
`25
`0.6
`65.6
`
`10
`0.5
`200
`8
`218.5
`
`13.12
`78.72
`
`2622
`2840.5
`
`12.70%
`38.11%
`
`0.35%
`0.02%
`
`WS Excipient
`max
`min
`
`WS Polymer Binder
`max
`min
`
`Second Disintegrant
`max
`min
`
`10
`0.5
`200
`0.6
`211.1
`
`42.22
`253.32
`
`10
`30
`25
`8
`73
`
`876
`949
`
`10
`0.5
`25
`8
`43.5
`
`8.7
`52.2
`
`10
`30
`200
`0.6
`240.6
`
`2887.2
`3127.8
`
`10
`0.5
`25
`0.6
`36.1
`
`10
`30
`200
`8
`248
`
`433.2
`469.3
`
`49.6
`297.6
`
`3.95%
`
`1.05%
`
`19.16%
`
`0.32%
`
`2.13%
`
`3.36%
`
`78.95%
`
`2.63%
`
`15.33%
`
`0.02%
`
`0.24
`78.96
`
`85.22
`2925.72
`
`0.76
`254.08
`
`28.47
`977.47
`
`0.16
`52.36
`
`93.83
`3221.63
`
`92.31%
`
`16.67%
`
`1.41
`470.71
`
`8.93
`306.53
`
`12.67%
`38.00%
`
`0.34%
`0.02%
`
`3.94%
`
`1.02%
`
`19.10%
`
`0.31%
`
`2.12%
`
`3.26%
`
`78.72%
`
`2.56%
`
`15.28%
`
`0.02%
`
`0.30%
`
`2.91%
`
`0.30%
`
`2.91%
`
`0.30%
`
`2.91%
`
`0.30%
`
`2.91%
`
`92.03%
`0.30%
`
`16.18%
`2.91%
`
`Par Pharm., Inc.
`Exhibit 1017
`Page 001
`
`