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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000002
`
`

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`WO 2008/056746
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000004
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`WO 2008/056746
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`DUK SAN NEOLUX
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`PAGE 000005
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`WO 2008/056746
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`DUK SAN NEOLUX
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`PAGE 000006
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`WO 2008/056746
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`PAGE 000007
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`
`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000008
`
`

`
`WO 2008/056746
`
`PCT/JP2007/071728
`
`[0029]
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`$73‘ ‘rx“fC(3) iii‘ Archiv der Pharmazie (Weinheim, Germany),1987,320(3),p280
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000009
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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000010
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`

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`WO 2008/056746
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`PCT/JP2007/071728
`
`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000011
`
`

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`WO 2008/056746
`
`827170I7002mTCP
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000012
`
`

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`WO 2008/056746
`
`827170I7002mTCP
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000013
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`PAGE 000014
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`WO 2008/056746
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`827170I7002mTCP
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`DUK SAN NEOLUX
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`PAGE 000015
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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000016
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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000017
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000018
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000019
`
`

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`WO 2008/056746
`
`PCT/JP2007/071728
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`[0042]
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`DUK SAN NEOLUX
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`PAGE 000020
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
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`PAGE 000021
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`[0048]
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000023
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000024
`
`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000025
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`[0061]
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000026
`
`

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`WO 2008/056746
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`PCT/JP2007/071728
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`[0067]
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000027
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`

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`WO 2008/056746
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`PCT/JP2007/071728
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`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000028
`
`

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`WO 2008/056746
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`PCT/JP2007/071728
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`24g (33.4H1moL HM:63.4%) %fi%7‘:o
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`APCHVIS, m/z 719 [M+1]+
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`fi§E)§,426°C
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`[0075]
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`H§Eéfi’”e%t%“sw%.?fiLf:20m1: E 7~?;<::c0:\ fi’E@§»\°~?~‘/“r7i\ (11) 0.071 g (0.32 mmol) \
`
`5?“/I/V (5 ml), W ten—7“7’wm%x74y 0. 32 m1(1.26 mmo1) $31302‘ 60°C‘? 30
`
`DUK SAN NEOLUX
`EXHIBIT 1017
`PAGE 000029
`
`

`
`WO 2008/056746
`
`PCT/JP2007/071728
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