WILLIAM R. ROUSH
`
`BIOGRAPHICAL DATA
`
`
`
`1974
`1977
`1977-1978
`
`Chula Vista, California, February 20, 1952
`
`BORN:
`
`EDUCATION:
`
`B. S., University of California, Los Angeles
`
`Ph. D., Harvard University
`
`Postdoctoral, Harvard University
`
`ACADEMIC POSITIONS:
`1978-1983
`
`Assistant Professor of Chemistry, M.I.T.
`1983-1987
`
`Associate Professor of Chemistry, M.I.T.
`1987-1989
`
`Associate Professor of Chemistry, Indiana University
`1989-1995
`
`Professor of Chemistry, Indiana University
`1995-1997
`
`Distinguished Professor of Chemistry, Indiana University
`1997-2005
`
`Warner Lambert/Parke-Davis Professor of Chemistry, Univ. of Michigan
`2002-2004
`
`Chair, Department of Chemistry, University of Michigan
`2005-2007
`
`Adjunct Professor of Chemistry, University of Michigan
`2005-present
`
`Professor of Chemistry, Scripps Research Institute (Florida)
`
`Executive Director of Medicinal Chemistry, Scripps Research Institute (FL) 2005-present
`
`Associate Dean of the Graduate Program, Scripps Research Institute (FL)
`2005-2016
`
`OTHER APPOINTMENTS:
`
`
`BioInformation Associates, Principal and Consultant
`1981-2001
`
`Genzyme Corporation, Consultant
`1983-1997
`
`Genzyme Corporation, Pharmaceuticals Division Board Member
`1994-1997
`
`NIH Medicinal Chemistry Study Section, Ad Hoc Member
`1984-1988
`
`Special NIH Study Sections, Ad Hoc Member
`1984-1988
`
`Chemtracts, Expert Analyst
`1986-1999
`
`Secretary-Treasurer, ACS Division of Organic Chemistry
`1990-1993
`
`Chairman, ACS Division of Organic Chemistry
`1995
`
`Alternate Councilor, ACS Division of Organic Chemistry
`1999-2002
`
`NIH Medicinal Chemistry Study Section, Member
`1990-1993
`
`Chairman, NIH Medicinal Chemistry Study Section
`1993-1995
`
`NIGMS Council, Ad-Hoc Member
`1998
`
`Editorial Board, Organic Reactions
`1991-2002
`
`Board of Directors, Organic Reactions
`1995-present
`
`Eli Lilly and Company, Consultant
`1991-present
`
`Editorial Board, Encyclopedia of Reagents for Organic Synthesis
`1992-2002
`
`Editorial Board, Organic Syntheses
`1993-2002
`
`Board of Directors, Organic Syntheses
`2003-present
`
`ArQule, Scientific Advisory Board Member
`1994-2003
`
`Consultant, NeXstar Pharmaceuticals, Inc.
`1994-1998
`
`Organizing Committee, NSF Workshop on
`
`
`Organic Synthesis and Natural Products Chemistry
`1995-1997
`
`Consultant, Proscript, Inc.
`1996-1998
`
`Consulting Editorial Board, Tetrahedron
`1996-2002
`
`Consultant, Parke Davis
`1998-2001
`
`Consultant, Pfizer
`2001-2013
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 1 of 39
`
`

`
`1999-2016
`1999-present
`2000-2002
`2001-2003
`2004-2005
`2005-2007
`2005-2010
`2005-2010
`2006-2015
`2007-2009
`2008-2009
`2008-2012
`2012-2015
`2015-present
`
`1974
`1974
`1981
`1981-1983
`1981-1984
`1982-1986
`1992
`1994
`1996
`1998
`1999
`2002
`2004
`2006
`2009
`
`Associate Editor, Journal of the American Chemical Society
`
`Editorial Advisory Board, Organic Letters
`
`Steering Committee, Challenges for the Chemical Sciences in the
`
`
`21st Century, National Research Council
`
`Invenux, Inc., Scientific Advisory Board Member
`
`Consultant, GMP-Immunotherapeutics
`
`Member, AAAS Nomination Selection Committee
`
`Editorial Advisory Board, Chemical Biology & Drug Design
`
`Editorial Advisory Board, Beilstein Journal of Organic Chemistry
`
`Lycera, Scientific Advisory Board
`
`Editorial Advisory Board, Accounts of Chemical Research
`
`Consultant, Heartland Sweetners, LLC
`
`Scientific Advisory Board, Sandler Center for Basic Research
`
`
`In Parasitic Diseases, University of California, San Francisco
`
`Scientific Advisory Board, Center for Discovery and Innovation
`
`
`in Parasitic Diseases, University of California, San Francisco
`
`Consultant, IMF Therapeutics
`
`
`HONORS AND AWARDS:
`
`B.S. in Chemistry, Summa Cum Laude
`
`Phi Beta Kappa
`
`Merck Faculty Development Award
`
`Eli Lilly Grantee
`
`Roger and Georges Firmenich Career Development Chair
`
`
`in Natural Products Chemistry (MIT)
`
`Fellow of the Alfred P. Sloan Foundation
`
`Alan R. Day Award of the Philadelphia Organic Chemist's Club
`
`Arthur C. Cope Scholar Award, American Chemical Society
`
`ACS Akron Section Award
`
`Merit Award, National Institute of General Medical Sciences
`
`Distinguished Faculty Achievement Award, University of Michigan
`
`Paul G. Gassman Distinguished Service Award,
`
`
`ACS Division of Organic Chemistry
`
`ACS Ernest Guenther Award in the Chemistry of Natural Products
`
`Fellow, American Association for the Advancement of Science
`
`Fellow, American Chemical Society
`
`
`
`March, 1992
`February, 1993
`November, 1993
`January, 1994
`April, 1994
`March, 1995
`April, 1995
`April, 1995
`April, 1995
`May, 1996
`April, 1999
`
`NAMED LECTURESHIPS
`Glaxo Lecturer, University of North Carolina
`Burkett Lecturer, DuPauw University
`Bristol-Myers Squibb Lecturer, Syracuse University
`Abbott Lecturer, University of California at Berkeley
`Syntex Lecturer, University of Colorado
`J. Clarence Karcher Lecturer, University of Oklahoma
`Warner Lambert Lecturer, Ohio State University
`SmithKline-Beecham Lecturer, University of Puerto Rico
`Wyeth-Ayerst/Penn Lecturer, University of Pennsylvania
`Convention Intercantonale Romande pour l'Enseignement
`
`du 3ème Cycle en Chimie (Switzerland)
`Bristol Myers Squibb Lecturer, Columbia University
`2
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 2 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`INVITED PARTICIPATION IN SYMPOSIA AND CONFERENCES:
`Lecturer, Symposium on Synthetic Methods and Processes, M.I.T.
`Lecturer, Frontiers in Organic Synthesis Symposium, U. Vermont
`Lecturer, Thirteenth Annual NSF Workshop on Organic Synthesis
`
`and Natural Products Chemistry
`
`Merck Lecturer, Swarthmore College
`Bristol Myers Squibb Lecturer, MIT
`Closs Lecturer, University of Chicago
`Bristol Myers Squibb Lecturer, Harvard University
`Organic Synthesis Lecturer, UC Irvine
`Organic Syntheses Distinguished Lecturer, Notre Dame
`Abbott Distinguished Lecturer, Abbott
`Novartis Lecturer, University of Texas, Austin
`Lilly Lecturer, University of Minnesota
`Frontiers in Chemistry Lecturer, Case Western Reserve
`American Cyanamid Lecturer, Bryn Mawr
`Bristol Myers Squibb Lecturer, Scripps Research Institute
`Ritchie Memorial Lecturer, Sydney Univ. Chemical Society,
`
`Sydney, Australia
`Boehringer-Ingelheim Lecturer, Université de Sherbrooke
`Bristol Myers Squibb Lecturer, University of Illinois
`Merck Lecturer, French Organic Chemical Society, Paris
`Oppolzer Lecturer, University of Geneva
`Servier Lecturer, Université de Montreal
`Pfizer Lecturer, Universitiy of Ottawa
`Pfizer Lectureship, Guelph-Waterloo Centre
`Roche Lecturer, University of Colorado, Boulder
`Gary Griffin Memorial Lecture, Univ. of New Orleans
`Pfizer Lecturer, Harvard University
`Boehringer Ingelheim Lecturer, University of Alberta
`Wyeth Lecturer, Princeton University
`AstraZeneca Lecture, University of British Columbia
`Bayer Lecture, University of Pennsylvania
`Merck Frosst Distinguished Lectureship, Queen’s University
`GlaxoSmithKline Lecturer, 6th Bristol Synthesis Meeting
`Donald Cram Lecturer, UCLA
`Ernst Schering Lecture, Berlin
`Robert Murray Lecture, University of Missouri
`Mack Award Lecture, Ohio State University
`Ireland Lecture, University of Virginia
`Robert A. Welch Lecture, Texas A&M University
`Robert A. Welch Lecture, Sam Houston State University
`Robert A. Welch Lecture, Texas Women’s University
`Molecular Basis of Disease Distinguished Lecturer,
`
`Georgia State University
`Organic Chemistry Frontiers Lecture, University of Hong Kong
`Eastman Lecture, University of California, Santa Barbara
`Regent Beth Fitzsimmons Lectureship, Eastern Michigan Univ.
`
`
`April, 1999
`February, 2000
`April, 2000
`April, 2000
`May, 2000
`October, 2000
`November, 2000
`March, 2001
`March, 2001
`April, 2001
`November, 2001
`December, 2001
`July, 2002
`November, 2002
`November, 2002
`March, 2003
`October, 2003
`November, 2003
`March, 2004
`June, 2004
`January, 2005
`February, 2005
`March, 2005
`September, 2005
`December, 2005
`February, 2006
`October, 2006
`December, 2006
`April, 2007
`November, 2007
`December, 2007
`March, 2008
`April, 2008
`October, 2008
`January, 2009
`January, 2009
`January, 2009
`January, 2014
`January, 2014
`April, 2014
`June, 2015
`
`1981
`1982
`1982
`
`3
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 3 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Conference on Yellow Rain, American Academy of Arts and Sciences,
`
`Cambridge, MA
`Lecturer, Advances in Applied Enzymology Symposium, M.I.T.
`Discussion Leader, Gordon Research Conference on Trichothecenes,
`
`Plymouth, NH
`Lecturer, Eli Lilly Organic Synthesis Symposium, Indianapolis, IN
`Lecturer, Federation of American Societies for Experimental Biology
`
`Conference on Trichothecenes, VT
`Lecturer, Spring Synthesis Symposium, Carleton University, Canada
`Lecturer, Gordon Research Conference on Trichothecenes and Fusarium
`
`Mycotoxins, Colby-Sawyer College, NH
`Lecturer, Gordon Research Conference on Carbohydrates, Tilton, NH
`Lecturer, ACS Symposium on Natural Products Synthesis
`
`(Metrochem '85), New York
`Lecturer, Ninth International Symposium on "Synthesis in Organic
`
`Chemistry", Oxford, England
`Lecturer, VPI Symposium on Latest Trends in Organic Synthesis,
`
`Blacksburg, VA
`Lecturer, Gordon Conference on Stereochemistry
`Lecturer, Federation of American Societies for Experimental Biology
`
`Conference on Trichothecene Mycotoxicosis, Colorado
`Lecturer, Molecular Recognition in Organic Synthesis Symposium,
`
`Ohio State University
`Keynote Lecturer, 25th Annual MIKIW Meeting, Lawrence, KA
`Lecturer, Symposium on "Asymmetric Synthesis of Carbohydrates from
`
`Acyclic Precursors," 194th National ACS Meeting, New Orleans
`Lecturer, Indiana University Chemistry Addition Dedication Symposium
`Lecturer, Philadelphia and Wilmington Organic Chemists Club 20th
`
`Biennial Symposium
`Lecturer, Symposium on Natural Products Synthesis, Southeast Regional
`
`ACS Meeting, Corpus Christi, TX
`Lecturer, Award Symposium for the 1990 ACS Award for Creative Work
`
`in Synthetic Organic Chemistry received by Clayton Heathcock,
`
`Boston ACS Meeting
`Lecturer, Symposium on Natural Products Synthesis, 23rd Great Lakes
`
`Regional ACS Meeting, DeKalb, IL
`Lecturer, U.S.-England NSF-SERC Workshop on Organic Synthesis,
`
`Pingree Park, Colorado
`Lecturer, "Organometallic Reagents in Carbohydrate Synthesis"
`
`Symposium, 1991 ACS Meeting in Atlanta
`Lecturer, "Current Methods for Enantioselective Synthesis," sponsored
`
`by Monsanto Company, St. Louis
`Lecturer, "Synthesis of Natural Products" Symposium, 24th Great Lakes
`
`Regional ACS Meeting, Indianapolis
`Lecturer, Gordon Conference on Reactions and Processes
`Lecturer, Symposium on Heterocycles in Asymmetric Synthesis,
`
`13th International Congress of Heterocyclic Chemistry, Corvallis
`Lecturer, Symposium on Natural Products Synthesis, SERMACS
`
`North Carolina
`Lecturer, Symposium on Asymmetric Processes, Royal Society
`
`of Chemistry Perkin Division Congress, Manchester, England
`Lecturer, 1992 Nozaki Conference, Yokohama, Japan
`4
`
`1983
`1983
`1983
`1983
`1984
`1985
`1985
`1985
`1985
`1985
`1986
`1986
`1986
`1987
`1987
`1987
`1988
`1988
`1988
`
`1990
`1990
`1990
`1991
`1991
`1991
`1991
`1991
`1991
`
`1992
`1992
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 4 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Lecturer, XVIth International Carbohydrate Symposium, Paris, France
`Award Lecture, 1992 Alan R. Day Award given by the
`
`Philadelphia Organic Chemist's Club
`Lecturer, VIIIth International Meeting on Boron Chemistry, Knoxville, TN
`Lecturer, 3rd Max Tschler Memorial Lecture Meeting,
`
`Kitasato Institute, Tokyo, Japan
`Lecturer, Award Symposium for the 1994 ACS Award for Creative Work
`
`in Synthetic Organic Chemistry received by Stuart Schreiber,
`
`San Diego National ACS Meeting
`Lecturer, Stereochemistry Gordon Conference, Newport, R.I.
`Award Lecture, 1994 Arthur C. Cope Award Symposium,
`
`Washington D.C. National ACS Meeting
`Lecturer, Symposium on Total Synthesis of Natural Products, 78th
`
`Canadian Society of Chemistry Conference, Guelph, Ontario
`Lecturer, Fifth International Meeting of the French-American Chemical
`
`Society, Bordeaux, France
`Lecturer, NSF Workshop on Organic Synthesis and Natural Products
`
`Chemistry, Tomales Bay, CA
`Lecturer, Princeton ACS Organic Chemistry Symposium
`Lecturer, Gulf Coast Chemistry Conference, Pensacola Beach, FL
`Lecturer, Symposium on Organometallics in Organic Transformations
`
`Synthesis and Asymmetric Catalysis, Pacific Basin Chemical
`
`Congress, Hawaii
`Lecturer, Symposium on Recent Advances in Organic Synthesis,
`
`University of Montreal
`Lecturer, NSF Workshop on Organic Synthesis and Natural Products
`
`Chemistry, Minary Conference Center, Squam Lake, NH
`Lecturer, Natural Products Gordon Conference
`Lecturer, Second Annual Procter & Gamble Pharmaceuticals
`
`Colloquium on Organic Synthesis
`Lecturer, 7th Brazilian Meeting on Organic Synthesis, Rio de Janeiro
`Lecturer, Lexington, KY, ACS Section Meeting
`Lecturer, Award Symposium for the 1997 ACS Hudson Award in
`
`Carbohydrate Chemistry, received by Samuel Danishefsky,
`
`San Francisco National ACS Meeting
`Lecturer, Symposium on the Art of Organic Synthesis, 80th
`
`Canadian Society of Chemistry Conference, Windsor, Ontario
`Lecturer, NSF Workshop on Organic Synthesis and Natural Products
`
`Chemistry, Tomales Bay, CA
`Lecturer, University of Colorado-Syntex/Roche Symposium on Organic
`
`Synthesis, Boulder, CO
`Lecturer, Natural Products Gordon Conference, New England College, NH
`Lecturer, Heterocycles Gordon Conference, Salve Regina University, RI
`Lecturer, Chemistry as a Life Science Symposium X - 2000, Rutgers
`Lecturer, Norvartis Lectureship Series
`Lecturer, Award Symposium for the 2000 ACS Ernest Guenther Award
`
`received by Pierre Potier, San Francisco National ACS Meeting
`Plenary Lecturer, Symposium on Organic Synthesis, Hope College
`Lecturer, AstraZeneca Excellence in Chemistry Award Symposium
`Lecturer, Advances in Asymmetric Synthesis Symposium,
`
`2000 International Chemical Congress of Pacific Basin
`
`Societies Meeting, Honolulu, Hawaii
`5
`
`1992
`1992
`1993
`1993
`1994
`
`1994
`1994
`
`1995
`1995
`1995
`1995
`1995
`1995
`
`1996
`1996
`1996
`1996
`
`1996
`1997
`1997
`
`1997
`1997
`
`1998
`1998
`1998
`2000
`2000
`2000
`
`2000
`2000
`
`2000
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 5 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Lecturer, 2nd Annual Connecticut Organic Chemistry Symposium
`Lecturer, 2nd Spring Organic Chemistry Symposium, North Jersey ACS
`Distinguished Alumni Lecture, Lilly Grantee Symposium
`Lecturer, Third International Symposium on New Synthetic Methods,
`
`sponsored by Sepracor, Florida
`Plenary Lecturer, Symposium on “Recent Advances in Synthetic
`
`Organic Chemistry,” Lilly Research Laboratories, Spain
`Plenary Lecturer, IUPAC Meeting on Organic Synthesis
`
`Christchurch, New Zealand
`Plenary Lecturer, XXIst International Carbohydrate Symposium,
`
`Cairns, Australia
`Lecturer, Reactions and Processes Gordon Conference, Rhode Island
`Lecturer, Carbohydrates Gordon Conference, New Hampshire
`Lecturer, 4th Annual UCSD/Merck Symposium on Perspectives
`
` in Organic Synthesis, UCSD
`Award Lecture, Guenther Award Symposium, ACS, Anaheim
`Lecturer, Symposium on Frontiers of Organic Synthesis and New
`
`Methodologies, ACS Central Regional Meeting, Indianapolis
`Lecturer, Natural Products Gordon Conference, New Hampshire
`Plenary Lecturer, ORCHEM 2004, Göttingen, Germany
`Plenary Lecturer, New Frontiers in Organic Synthesis Symposium,
`
`Lilly-Spain (Madrid)
`Keynote Speaker, Singapore International Chemical Conference, Singapore
`Plenary Speaker, 9th Frank Warren Conference on Organic Chemistry
`
`University of Cape Town, South Africa
`Lecturer, Frontiers in Biomedical Research Symposium, Indian Wells, CA
`Lecturer, Florida Annual Meeting and Exposition (FAME), Orlando
`Lecturer, Fresnius Award Symposium, ACS, Chicago
`Lecturer, 11th ICSN Symposium, Gif-sur-Yvettte, France
`Lecturer, ACS Advances in Drug Design Symposium, San Francisco
`Lecturer, Balticum Organicum Syntheticum, Vilnius, Lithuania
`Lecturer, Heterocycles Gordon Conference, Newport, Rhode Island
`Lecturer, Donald S. Matteson Symposium in Organic Chemistry,
`
`Washington St. University
`Plenary Lecturer, Eli Lilly Europe Graduate Student Awards Symposium
`
`(Madrid)
`Lecturer, Natural Products Gordon Conference
`Lecturer, Beckmann Symposium on New Frontiers in Academic
`
`Medicine and Therapeutic Development, City of Hope, Los Angeles
`Lecturer, Symposium on Drug Design, Discovery and Delivery
`
`University of Central Florida, Tampa
`Plenary Lecturer, 11th Annual Florida Heterocyclic and Synthetic
`
`Conference, Gainesville, FL
`Lecturer, New York Academy of Sciences Symposium on “Metabolic
`
`Regulation and Human Disease”
`Lecturer, Robert B. Woodward Symposium, ACS, Boston
`Lecturer, 11th Biennial Frontiers in Organic Chemistry Symposium,
`
`University of Illinois (sponsored by Johnson and Johnson)
`Plenary Lecturer, Eckerd College Science Symposium, Exploring
`
`Critical Issues in Science”
`Plenary Lecturer, Symposium on Natural Products Synthesis,
`
`Organic Chemistry Division of the Korean Chemical Society,
`6
`
`2001
`2001
`2002
`2002
`2002
`2002
`2002
`2003
`2003
`2003
`2004
`2004
`2004
`2004
`2005
`2005
`2006
`2006
`2006
`2007
`2007
`2007
`2008
`2008
`2008
`2008
`2009
`2009
`2009
`2010
`2010
`2010
`2010
`2010
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 6 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`SEMINARS AT UNIVERSITIES AND RESERCH INSTITUTES:
`Massachusetts Institute of Technology
`Wesleyan University
`Duke University
`California Institute of Technology
`University of Pennsylvania
`University of Virginia
`University of Chicago
`Brown University
`S.U.N.Y., Stony Brook
`Northeastern University
`Yale University
`Cornell University
`S.U.N.Y., Buffalo
`University of California, Berkeley
`Rensselaer Polytechnic Institute
`University of Rochester
`Hunter College
`University of Illinois, Urbana-Champaign
`Brandeis University
`Harvard University
`University of Pittsburgh
`
`Jeju, Korea
`
`Lecturer, 4th PKU-Eli Lilly Symposium of Organic Chemistry,
`
`Peking University, China
`Plenary Lecturer, Zing Conference on Natural Products Synthesis
`
`and Biosynthesis, Lanzarote, Canary Islands
`Lecturer, National Organization for the Professional Advancement of
`
`Black Chemists and Chemical Engineers Symposium, San Diego
`Lecturer, National Medicinal Chemistry Symposium, Tuscon, AR
`Lecturer, Victor Grignard Nobel Centenial-ACS Chemical
`
`Breakthrough Award Symposium, Lyon, France
`Lecturer, Heterocycles Gordon Conference, Salve Regina College, RI
`Lecturer, SERMACS Chemical Biology Symposium, Raleigh, NC
`Lecturer, National Organic Symposium, Seattle
`Plenary Lecturer 24th International Society of Heterocyclic Chemistry,
`
`Shanghai, China
`Lecturer, Stereochemistry Gordon Conference, Salve Regina College, RI
`Keynote Lecture, 8th Singapore International Chemical Conference
`
`(SICC-8)
`Keynote Lecturer, Organic Synthesis Symposium, Florida ACS
`
`Organic Division
`Lecturer, Symposium on Interface of Science and Technology as
`
`Applied to Natural Product Research, Budapest, Hungary
`Keynote Lecturer, Eli Lilly Grantee Symposium
`
`Indianapolis, IN
`Lecturer, 6th Pharmaron Symposium, Beijing, China
`
`
`2011
`2011
`2012
`2012
`2012
`2012
`2012
`2012
`2013
`2013
`2014
`2014
`2015
`2015
`2016
`2016
`
`May, 1977
`March, 1980
`March, 1980
`March, 1981
`September, 1981
`February, 1982
`November, 1982
`November, 1982
`November, 1982
`November, 1982
`February, 1983
`March, 1983
`September, 1983
`April, 1984
`April, 1984
`May, 1984
`October, 1984
`November, 1984
`February, 1985
`March, 1985
`March, 1985
`
`7
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 7 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`University of West Virginia
`Pennsylvania State University
`Columbia University
`Cambridge University, Cambridge, England
`University of Zurich, Switzerland
`University of Massachusetts, Amherst
`Boston University
`Indiana University
`Michigan State University
`Brandeis University
`Purdue University
`Indiana University
`Texas A&M
`New York Academy of Sciences
`University of Texas, Austin
`Indiana University-Purdue University at Indianapolis
`University of Illinois, Urbana-Champaign
`University of Louisville
`University of Pennsylvania
`University of Minnesota
`University of North Dakota
`University of South Carolina
`Emory University
`Case Western Reserve University
`University of Tennessee
`Boston University
`University of Akron
`S.U.N.Y., Stony Brook
`Northwestern University (2 lectures)
`University of Wisconsin
`Scripps Research Institute, La Jolla, CA
`University of Rochester
`University of Michigan
`University of Montreal, Canada
`Tohoku University (Sendai)
`University of Tokyo
`Kyoto University
`Okayama University of Science
`Nagoya University
`Miami University, Ohio
`Massachusetts Institute of Technology
`Colorado State University
`Yale University
`Notre Dame
`Harvard University
`Hope College
`Calvin College
`University of Maryland
`University of Nebraska
`University of Missouri, Columbia
`Okayama University of Science
`Waseda University (Tokyo)
`
`8
`
`March, 1985
`October, 1985
`November, 1985
`January, 1986
`January, 1986
`February, 1986
`March, 1986
`April, 1986
`April, 1986
`May, 1986
`May, 1986
`June, 1986
`August, 1986
`November, 1986
`December, 1988
`February, 1989
`February, 1989
`March, 1989
`February, 1990
`February, 1990
`February, 1990
`November, 1990
`November, 1990
`February, 1991
`February, 1991
`March, 1991
`April, 1991
`May, 1991
`July, 1991
`November, 1991
`November, 1991
`February, 1992
`March, 1992
`March, 1992
`May, 1992
`May, 1992
`May, 1992
`May, 1992
`May, 1992
`September, 1992
`September, 1992
`September, 1992
`October, 1992
`December, 1992
`January, 1993
`February, 1993
`February, 1993
`February, 1993
`April, 1993
`April, 1993
`October, 1993
`October, 1993
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 8 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Tokyo Institute of Technology
`Keio University (Tokyo)
`Boston College
`Stanford University
`University of California at Berkeley
`Bucknell University
`University of Pittsburgh
`Wayne State University
`University of Texas, Austin
`Texas A&M University
`University of Minnesota
`University of California at Irvine
`California Institute of Technology
`University of California at San Francisco
`University of California, San Diego
`Rensselaer Polytechnic Institute
`University of Michigan
`University of Toronto
`University of Utah
`Université de Neuchâtel, Switzerland
`Université de Fribourg, Switzerland
`Université de Lausanne, Switzerland
`Université de Genève, Switzerland (2 lectures)
`Université de Paris-Sud, Orsay, France
`University of Illinois, Chicago Circle
`University of Akron
`Brandeis University
`University of Rochester
`Iowa State University
`University of Virginia
`University of Kentucky
`Louisiana State University
`Hunter College
`Michigan St. University
`North Carolina State University
`University of Michigan (Dept. of Biological Chemistry)
`University of Toledo
`Columbia University
`Swarthmore College
`University of Arkansas
`University of Michigan (Biophysics Research Division)
`University of Pennsylvania
`University of Arizona
`University of Notre Dame
`Ohio State University
`Stanford University
`Memorial Sloan Kettering
`Texas A&M University
`Colorado St. University
`Boston College
`University of Maryland
`Purdue University
`
`9
`
`October, 1993
`October, 1993
`October, 1993
`January, 1994
`January, 1994
`March, 1994
`March, 1994
`April, 1994
`March, 1995
`March, 1995
`April, 1995
`November, 1995
`November, 1995
`November, 1995
`January, 1996
`February, 1996
`March, 1996
`April, 1996
`April, 1996
`May, 1996
`May, 1996
`May, 1996
`May, 1996
`May, 1996
`October, 1996
`November, 1996
`February, 1997
`March, 1997
`March, 1997
`March, 1997
`April, 1997
`September, 1997
`November, 1997
`April, 1998
`November, 1998
`March, 1999
`April, 1999
`April, 1999
`April, 1999
`October, 1999
`October, 1999
`November, 1999
`May, 2000
`October, 2000
`November, 2000
`January, 2001
`February, 2001
`November, 2001
`January, 2002
`March, 2002
`April, 2002
`April, 2002
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 9 of 39
`
`

`
`February, 2003
`Wayne St. University
`March, 2003
`Université de Rene, France
`March, 2003
`University of Marseille, France
`March, 2003
`University de Lyon, France
`March, 2004
`California Institute of Technology
`January, 2005
`Florida St. University, Tallahassee
`January, 2006
`University of Cape Town, South Africa
`February, 2006
`University of Florida, Gainesville
`April, 2006
`Wellesley College
`April, 2006
`Rutgers University
`April, 2006
`Georgia Tech, Atlanta
`April, 2006
`SUNY Buffalo
`April, 2007
`University of Central Florida
`December, 2007
`Technical University, Berlin
`April, 2008
`Oregon St. University
`April, 2008
`Ohio State University
`April, 2009
`Northwestern University
`May, 2009
`University of Wisconsin
`November, 2009
`Rollins College, Tampa FL
`April, 2010
`University of Arizona, Tucson
`September, 2010
`University of Florida, Gainesville
`October, 2010
`Virginia Tech, Blacksburg VA
`March, 2011
`University of South Florida, Tampa, FL
`April, 2011
`Seoul National University, Seoul, Korea
`April, 2011
`Yonsei University, Daejeon, Korea
`April, 2011
`Korean Institute of Chemical Technology, Daejeon, Korea
`November, 2011
`LSU, Baton Rouge, LA
`January, 2012
`University of California, Irvine
`April, 2012
`Shanghai Institute of Organic Chemistry, China
`April, 2012
`National University of Singapore, Singapore
`University of Michigan Center for Discovery of New Medicines November, 2013
`University of Toledo
`November, 2013
`Chinese University of Hong Kong
`January, 2014
`Hong Kong University of Science and Technology
`January, 2014
`Scripps Research Institute, La Jolla, CA
`January, 2016
`University of Florida, Gainesville
`February, 2016
`California State University, Fullerton
`February, 2016
`
`
`
`* * * * * * * * * * *
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`February, 1977
`February, 1977
`May, 1979
`March, 1980
`September, 1980
`October, 1980
`October, 1980
`
`10
`
`SEMINARS AT COMPANIES:
`Merck, Rahway
`Pfizer, Groton
`Ciba-Geigy Pharmaceutical, Summit
`DuPont, Wilmington
`Shell Development Co., Modesto, CA
`BASF Wyandotte Corporation
`Warner-Lambert/Parke-Davis
`
`
`
`
`
`
`
`
`
`
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 10 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Bristol Laboratories, Syracuse
`Merck, Rahway
`Squibb Institute for Medical Research
`Lederle Laboratories, Pearl River NY
`Burroughs-Wellcome, Research Triangle
`Merck, West Point
`Eli Lilly, Indianapolis
`Sandoz Pharmaceuticals, East Hanover, NJ
`Pfizer, Groton
`Abbott Laboratories, Chicago
`Rohm & Haas, Philadelphia
`Eli Lilly, Indianapolis
`Upjohn Pharmaceutical Company, Kalamazoo
`Sterling-Winthrop Research Institute
`American Cyanamide, Princeton
`Firmenich SA, Geneva, Switzerland
`Stuart Pharmaceuticals, Wilmington
`Exxon Research and Engineering Co., NJ
`Squibb Institute for Medical Research, Princeton
`E. R. Squibb Company, New Brunswick, NJ
`Revlon Health Care Group, Tuckahoe, NY
`Hoffmann-La Roche & Co., Basel, Switzerland
`Schering Corporation, Bloomfield, NJ
`Smith Kline & French, Philadelphia
`DuPont, Wilmington
`Proctor & Gamble, Cincinnati
`Genzyme Fine Chemicals, Haverhill, England
`Upjohn, Kalamazoo
`Rohm & Haas, Philadelphia
`Wyeth-Ayerst, Philadelphia
`Berlex, New Jersey
`E. R. Squibb Company, New Brunswick
`Boehringer Ingelheim, Connecticut
`Lederle Laboratories, Pearl River, NY
`Eli Lilly, Indianapolis
`Merck, Rahway
`Janssen Research Foundation, Spring House, PA
`Genzyme Corporation, Boston, MA
`American Cyanamide, Princeton, NJ
`Anaquest, NJ
`BioMega, Montreal, Canada
`Hoffmann La Roche, Nutley, NJ
`Sankyo (Shinagawa, Tokyo)
`Suntory Institute (Osaka, Japan)
`Smith Kline Beecham, England
`DuPont Merck, Wilmington
`Sterling Winthrop Research Institute, Albany, NY
`Eli Lilly, Tippicanoe Laboratories
`Burroughs Wellcome, North Carolina
`Abbott Laboratories (Process Chemistry)
`Kao Corporation, Japan
`RIKEN Institute, Tokyo, Japan
`
`11
`
`December, 1980
`February, 1981
`February, 1981
`May, 1981
`May, 1981
`October, 1981
`October, 1981
`November, 1981
`November, 1981
`May, 1982
`September, 1983
`March, 1984
`March, 1984
`April, 1984
`May, 1984
`May, 1984
`October, 1984
`March, 1985
`May, 1985
`May, 1985
`November, 1985
`January, 1986
`March, 1986
`September, 1986
`March, 1987
`October, 1987
`January, 1988
`March, 1988
`October, 1988
`March, 1989
`May, 1989
`February, 1990
`March, 1990
`May, 1990
`June, 1990
`May, 1991
`June, 1991
`October, 1991
`January, 1992
`January, 1992
`March, 1992
`May, 1992
`May, 1992
`May, 1992
`July, 1992
`September, 1992
`October, 1992
`January, 1993
`May, 1993
`September, 1993
`September, 1993
`October, 1993
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 11 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Abbott Laboratories (Discovery Chemistry)
`May, 1994
`NeXagen, Boulder, Colorado
`May, 1994
`Eli Lilly, Indianapolis
`June, 1994
`Agouron Pharmaceuticals, San Diego
`November, 1994
`Zeneca Pharmaceuticals Group, Wilmington, DE
`November, 1994
`Warner Lambert (Parke Davis), Ann Arbor, MI
`April, 1995
`Wyeth-Ayerst, Princeton, NJ
`April, 1995
`Ligand Pharmaceuticals, San Diego
`May, 1995
`Pfizer, Groton, CT
`May 1995
`Mont-Saint-Guibert Development Center (Lilly), Brussels, Belgium
`June, 1995
`Merck-Frosst, Montreal
`September, 1995
`Merck, Rahway
`April, 1996
`Merck, West Point
`April, 1996
`CNRS, Gif sur Yvette, France
`May, 1996
`Abbott Laboratories (Process Chemistry)
`May, 1997
`Wyeth Ayerst (Lederle Laboratories)
`November, 1997
`Merck, Rahway
`November, 1997
`Warner Lambert (Parke Davis), Ann Arbor, MI
`February, 1998
`Warner Lambert (Parke Davis; Biochem. Department)
`April, 1998
`Novartis, Summit, NJ
`December, 1998
`Tularik, San Francisco, CA
`January, 1999
`RW Johnson, Spring House, PA
`February, 1999
`Ligand Pharmaceuticals, San Diego, CA
`May, 1999
`RW Johnson, Rariton, NJ (Process Research)
`October, 1999
`Sepracor, Marlborough, MA
`November, 1999
`Warner Lambert (Parke Davis), Holland, MI
`January, 2000
`Schering Plough Research Institute, NJ
`March, 2000
`Dow AgroSciences, Midland, MI
`September, 2000
`Goodyear, Akron, OH
`April, 2001
`Pfizer, Groton
`June, 2001
`RW Johnson, San Diego
`January, 2002
`Bristol Myers Squibb, Princeton, NJ
`February, 2002
`Pharmacia (Kalamazoo, MI)
`September, 2002
`Seattle Genetics (Seattle, WA)
`September, 2002
`Pharmacia (Skokie, IL)
`November, 2002
`Boehringer-Ingelheim, Montreal
`November, 2002
`Pharmacia (St. Louis)
`January, 2003
`Celera (San Francisco)
`April, 2003
`Merck, San Diego
`April, 2003
`Array BioPharma (Boulder, CO)
`September, 2003
`Eli Lilly, MSG, Belguim
`October, 2003
`Hoffmann-La Roche, New Jersey
`November, 2003
`Merck, Rahway
`November, 2003
`Dow AgroSciences, Indianapolis
`September, 2004
`Amgen, Thousand Oaks, CA
`September, 2004
`Givaudan, Cincinnati
`February, 2005
`Bristol Meyers Squibb, New Brunswick, NJ
`March, 2005
`Wyeth-Ayerst Pharmaceuticals
`December, 2005
`Boheringer Ingelheim, CT
`April, 2006
`Pfizer, Technology Research Center, Cambridge, MA
`August, 2006
`Eli Lilly, Erl Wood, UK
`November, 2006
`Sanofi-Aventis, Frankfurt, Germany
`November, 2006
`
`12
`
`NOVARTIS EXHIBIT 2094
`Par v Novartis, IPR 2016-00084
`Page 12 of 39
`
`

`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`
`Merck Frosst, Montreal, Canada
`Tripos, Bude, UK
`GlaxoSmithKline, Harlow, UK
`GlaxoSmithKline, Stevenege, UK
`AstraZeneca, Waltham, MA
`Johnson & Johnson, San Diego
`Bristol Myers Squibb