`_________________________________
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`BEFORE THE PATENT TRIAL AND APPEAL BOARD
`_________________________________
`
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`NOVEN PHARMACEUTICALS, INC.,
`Petitioner
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`v.
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`NOVARTIS AG AND LTS LOHMANN THERAPIE-SYSTEME AG,
`Patent Owners
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`_________________________________
`
`
`Inter Partes Review No.: 2014-00550
`U.S. Patent No. 6,335,031
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`PETITIONER’S EXHIBIT LIST 1
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`Pursuant to 37 C .F.R. §42.63(e), Petitioner Noven submits the following
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`current exhibit list.
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`US. Patent No. 6,335,031, issued January 1, 2002
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`UK Patent Application GB 2,203,040 A, to Enz, published October
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`12, 1988 (“Enz”)
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`Handbook of Pharmaceutical Excipients, A- Wade and P. J. Weller
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`(eds.) 1994, 2nd Edition, The Pharmaceutical Press London (the
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`“Handbook”)
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`
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`Japanese Patent Application Publication No. JP 59-18412] to
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`Sasaki et al., published October 19, 1984
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`Certified English Translation of Japanese Patent Application
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`Publication No. JP 59-184121 to Sasaki et al. (“Sasaki”)
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`PCT Publication No. WO 95/024172 to Ebert et al, published
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`September 14, 1995 (“Ebert”)
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`Carey & Sundberg, ADVANCED ORGANIC CHEMISTRY, Part
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`A: Structure and Mechanism, 3rd Edition (Plenum Press, NY), pp.
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`
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`651-727 (1990)
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`Ex. 1008 U.S. Patent 4,948,807 (“Rosin”)
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`Ex. 1009 Elmalem et al. 1991, Neuropharmacology 30: 1059-1064
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`(“Elmalem”)
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`Ex. 1010 Declaration of Agis Kydonieus, Ph.D.
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`Ex. 1011 Declaration of Christian Schöneich, Ph.D.
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`Ex. 1012 “Safety/Tolerability Trial of SDZ ENA 713 in Patients with
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`Probable Alzheimer’s Disease,” John J. Sramek et al., Life
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`Sciences, Vol. 58, No. 15, pp. 1201-1207 (1996) (“Sramek”)
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`Ex. 1013 “New acetylcholinesterase inhibitor shows promise in largest
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`Alzheimer’s trial to date,” Formulary, Vol. 32, Dec. 1997
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`(“Formulary Article”)
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`Ex. 1014 ICH Topic Q 1 A, Stability Testing Guidelines: Stability Testing
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`of New Drug Substances and Products (CPMP/ICH/380/95)
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`Ex. 1015 Connors, Amidon, & Stella, Oxidation and Photolysis in Chemical
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`Stability of Pharmaceuticals – A Handbook for Pharmacists (2nd
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`Edition), John Wiley & Sons, NY (1986), pp. 82-114
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`2
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`Ex. 1016 Howard C. Ansel, Introduction to Pharmaceutical Dosage Forms,
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`4th Edition, Lea & Febiger, Philadelphia (1985), pp. 83-116
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`Ex. 1017 Ho-Leung Fung, Chapter 7 – Chemical Kinetics and Drug Stability
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`in MODERN PHARMACEUTICS (G.S. Banker and C.T. Rhodes,
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`eds.), Marcel Dekker, NY (1979), pp. 227-62
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`Ex. 1018 Miguel-Hidalgo, J., 2000, Current Opinion in CPNS Investigations
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`Drugs, 2000 2(4):438-453
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`Ex. 1019 Boccardi G. et al. Photochemical Iron(III)-Mediated Autoxidation
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`of Dextromethorphan. Chemical & Pharmaceutical Bulletin. Vol.
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`37, 308–310 (1989)
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`Ex. 1020 Bateman, L., Olefin Oxidation, Quarterly Review (1954) Vol. 8,
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`pp. 147–167
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`Ex. 1021 Linnell, R.H., The Oxidation of Nicotine. I. Kinetics of the Liquid
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`Phase Reaction Near Room Temperature. Tobacco Science, Vol.
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`4, pp. 89–91 (1960)
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`Ex. 1022 Resume/Curriculum Vitae of Agis Kydonieus, Ph.D.
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`Ex. 1023 Resume/Curriculum Vitae of Christian Schöneich, Ph.D.
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`3
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`Ex. 1024 U.S. Patent No. 5,602,176, issued Feb. 11, 1997
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`Ex. 1025 Redacted Copy of Bench Trial Transcript (Day 1). C.A. No. 13-
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`527, D.I. 154 (D. Del).
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`Ex. 1026 Redacted Copy of Bench Trial Transcript (Day 2). C.A. No. 13-
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`527, D.I. 155 (D. Del).
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`Ex. 1027 Redacted Copy of Bench Trial Transcript (Day 3). C.A. No. 13-
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`527, D.I. 156 (D. Del).
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`Ex. 1028 U.S. Patent No. 5,061,480. [Not Filed]
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`Ex. 1029 Transcript of 1/13/2015 Deposition of Dr. Agis Kydonieus
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`4
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`Dated: January 20, 2015
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`Respectfully submitted,
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`/Steven J. Lee/
`Steven J. Lee (Reg. No. 31,272)
`Michael K. Levy (Reg. No. 40,699)
`KENYON & KENYON LLP
`One Broadway
`New York, NY 10004-1007
`Tel: 212-425-7200
`Fax: 212-425-5288
`Counsel for Petitioner Noven Pharmaceuticals,
`Inc.
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`CERTIFICATE OF SERVICE
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` I
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` certify pursuant to 37 C.F.R. §42.6(e) that a copy of Noven’s current
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`Exhibit List and copies of Exhibits 1025, 1026, 1027, and 1028, were served by
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`hand on January 13, 2015 to Charlotte C. Jacobsen, Esq., of Fitzpatrick, Cella,
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`Harper & Scinto, 1290 Avenue of the Americas, New York, NY 10104-3800,
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`pursuant to 37 C.F.R. §42.63(e) and §42.53(f)(3). I also certify pursuant to 37
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`C.F.R. §42.6(e) that a copy the foregoing Exhibit List 1 and copies of Exhibits
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`1025, 1026, 1027, 1028 and 1029, were served electronically on January 20, 2015
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`pursuant to 37 C.F.R. §42.63(e) to counsel for Patent Owners at the following
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`email address: ExelonPatchIPR@fchs.com.
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`Dated: January 20, 2015
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`/Christopher J. Coulson/
`Christopher J. Coulson (Reg. No. 61,771)
`KENYON & KENYON LLP
`One Broadway
`New York, NY 10004-1007
`Tel: 212-425-7200
`Fax: 212-425-5288
`Counsel for Petitioner Noven Pharmaceuticals,
`Inc.
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